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TargetPhospholipase A2 group V
LigandBDBM50366784
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1764264 (CHEMBL4199511)
IC50 2200±n/a nM
Citation Giordanetto, FKnerr, LNordberg, PPettersen, DSelmi, NBeisel, HGde la Motte, HMånsson, ÅDahlström, MBroddefalk, JSaarinen, GKlingegård, FHurt-Camejo, ERosengren, BWikström, JWågberg, MBrengdahl, JRohman, MSandmark, JÅkerud, TRoth, RGJansen, FAhlqvist, M Design of Selective sPLA ACS Med Chem Lett9:600-605 (2018) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Phospholipase A2 group V
Name:Phospholipase A2 group V
Synonyms:PA2G5_HUMAN | PLA2G5 | Phospholipase A2 group V | Secretory phospholipase A2, group V (sPLA2-V)
Type:Protein
Mol. Mass.:15682.61
Organism:Homo sapiens (Human)
Description:n/a
Residue:138
Sequence:
MKGLLPLAWFLACSVPAVQGGLLDLKSMIEKVTGKNALTNYGFYGCYCGWGGRGTPKDGT
DWCCWAHDHCYGRLEEKGCNIRTQSYKYRFAWGVVTCEPGPFCHVNLCACDRKLVYCLKR
NLRSYNPQYQYFPNILCS
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BDBM50366784
n/a
NameBDBM50366784
Synonyms:CHEMBL4171084
TypeSmall organic molecule
Emp. Form.C19H15F3N2O4
Mol. Mass.392.3286
SMILESNC(=O)c1cc2ccc(OC(F)(F)F)cc2n1-c1cccc(CCC(O)=O)c1
Structure
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