Reaction Details |
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Target | Melatonin receptor type 1C |
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Ligand | BDBM50470866 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_104755 (CHEMBL712438) |
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Ki | 29±n/a nM |
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Citation | Mathé-Allainmat, M; Gaudy, F; Sicsic, S; Dangy-Caye, AL; Shen, S; Brémont, B; Benatalah, Z; Langlois, M; Renard, P; Delagrange, P Synthesis of 2-amido-2,3-dihydro-1H-phenalene derivatives as new conformationally restricted ligands for melatonin receptors. J Med Chem39:3089-95 (1996) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Melatonin receptor type 1C |
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Name: | Melatonin receptor type 1C |
Synonyms: | CKB | MTR1C_CHICK | Mel-1C-R | Mel1c receptor | Melatonin receptor type 1C |
Type: | PROTEIN |
Mol. Mass.: | 38595.98 |
Organism: | Gallus gallus |
Description: | ChEMBL_104739 |
Residue: | 346 |
Sequence: | MERPGSNGSCSGCRLEGGPAARAASGLAAVLIVTIVVDVLGNALVILSVLRNKKLRNAGN
IFVVSLSVADLVVAVYPYPLILSAIFHNGWTMGNIHCQISGFLMGLSVIGSIFNITAIAI
NRYCYICHSLRYDKLFNLKNTCCYICLTWTLTVVAIVPNFFVGSLQYDPRIYSCTFAQTV
STSYTITVVVVHFIVPLSIVTFCYLRIWILVIQVKHRVRQDCKQKIRAADIRNFLTMFVV
FVLFAVCWGPLNFIGLAVSINPSKVQPHIPEWLFVLSYFMAYFNSCLNAVIYGLLNQNFR
KEYKRILLMLRTPRLLFIDVSKGGTEGLKSKPSPAVTNNNQAEIHL
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BDBM50470866 |
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n/a |
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Name | BDBM50470866 |
Synonyms: | CHEMBL320810 |
Type | Small organic molecule |
Emp. Form. | C15H15NO |
Mol. Mass. | 225.2857 |
SMILES | CC(=O)NC1Cc2cccc3cccc(C1)c23 |
Structure |
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