| Reaction Details |
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 | Report a problem with these data |
| Target | Reverse transcriptase |
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| Ligand | BDBM50478032 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_601567 (CHEMBL1047747) |
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| IC50 | <10.0±n/a nM |
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| Citation |  Prajapati, DG; Ramajayam, R; Yadav, MR; Giridhar, R The search for potent, small molecule NNRTIs: A review. Bioorg Med Chem17:5744-62 (2009) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Reverse transcriptase |
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| Name: | Reverse transcriptase |
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| Synonyms: | n/a |
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| Type: | Protein |
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| Mol. Mass.: | 29598.37 |
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| Organism: | Human immunodeficiency virus 1 |
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| Description: | Q9WKE8 |
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| Residue: | 254 |
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| Sequence: | PISPITVPVKLKPGMDGPKVKQWPLTEEKIKALTEICTEMEKEGKIEKIGPENPYNTPVF
AIKKKDSTKWRKVVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLD
KDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIY
QYMDDLYVGSDLEIEQHRAKIEELRQHLLRWGFTTPDKKHQKEPPFLWMGYELHPDKWTV
QPIVLPEKDSWTVN
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| BDBM50478032 |
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| n/a |
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| Name | BDBM50478032 |
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| Synonyms: | CHEMBL275658 | GW4511 | GW564511 | GW69564 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H17ClF4N2O5S |
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| Mol. Mass. | 544.903 |
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| SMILES | Cc1cc(ccc1NC(=O)COc1ccc(Cl)cc1C(=O)c1cc(F)cc(c1)C(F)(F)F)S(N)(=O)=O |
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| Structure | 
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