| Reaction Details |
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 | Report a problem with these data |
| Target | Group 10 secretory phospholipase A2 |
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| Ligand | BDBM50040458 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_156341 (CHEMBL759984) |
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| IC50 | 380±n/a nM |
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| Citation |  Beaton, HG; Bennion, C; Connolly, S; Cook, AR; Gensmantel, NP; Hallam, C; Hardy, K; Hitchin, B; Jackson, CG; Robinson, DH Discovery of new non-phospholipid inhibitors of the secretory phospholipases A2. J Med Chem37:557-9 (1994) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Group 10 secretory phospholipase A2 |
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| Name: | Group 10 secretory phospholipase A2 |
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| Synonyms: | Group X secretory phospholipase A2 | PA2GX_HUMAN | PLA2G10 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 18153.11 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1442449 |
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| Residue: | 165 |
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| Sequence: | MGPLPVCLPIMLLLLLPSLLLLLLLPGPGSGEASRILRVHRRGILELAGTVGCVGPRTPI
AYMKYGCFCGLGGHGQPRDAIDWCCHGHDCCYTRAEEAGCSPKTERYSWQCVNQSVLCGP
AENKCQELLCKCDQEIANCLAQTEYNLKYLFYPQFLCEPDSPKCD
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| BDBM50040458 |
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| n/a |
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| Name | BDBM50040458 |
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| Synonyms: | (S)-4-((S)-(E)-Dec-3-enoylamino)-5-(naphthalen-2-ylsulfanyl)-pentanoic acid | CHEMBL152402 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H33NO3S |
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| Mol. Mass. | 427.599 |
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| SMILES | CCCCCC\C=C\CC(=O)N[C@@H](CCC(O)=O)CSc1ccc2ccccc2c1 |
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| Structure | 
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