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TargetTubulin polymerization-promoting protein
LigandBDBM50099946
Substrate/Competitorn/a
Meas. Tech.ChEMBL_925239 (CHEMBL3073731)
EC50>100000±n/a nM
Citation Young, DHTice, CMMichelotti, ELRoemmele, RCSlawecki, RARubio, FMRolling, JA Structure-activity relationships of phenylcyclohexene and biphenyl antitubulin compounds against plant and mammalian cells. Bioorg Med Chem Lett11:1393-6 (2001) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Tubulin polymerization-promoting protein
Name:Tubulin polymerization-promoting protein
Synonyms:25 kDa brain-specific protein | TPPP | TPPP_BOVIN
Type:PROTEIN
Mol. Mass.:23484.86
Organism:Bos taurus
Description:ChEMBL_106635
Residue:218
Sequence:
MADSRPKPANKTPPKSPGEPAKDKAAKRLSLEAEGAGEGAAAAGAELSALEEAFRKFAVH
GDARASGREMHGKNWSKLCRDCQVIDGRSVTVTDVDIVFSKIKGKSCRTITFEQFKEALE
ELAKKRFKDKSAEEAVREVHKLIEGKAPIISGVTKAISSPTVSRLTDTSKFTGSHKERFD
PSGRGKGRAGRVDLVDESGYVPGYKHAGTYDQKVQGGK
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  Blast E-value cutoff:
BDBM50099946
n/a
NameBDBM50099946
Synonyms:1,2,3-Trimethoxy-4-(6-nitro-cyclohex-3-enyl)-benzene | CHEMBL283411
TypeSmall organic molecule
Emp. Form.C15H19NO5
Mol. Mass.293.3151
SMILESCOc1ccc(C2CC=CC[C@H]2[N+]([O-])=O)c(OC)c1OC |c:8|
Structure
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