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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | D(1B) dopamine receptor | ||
| Ligand | BDBM50004822 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEMBL_1991503 (CHEMBL4625238) | ||
| Ki | 0.500000±n/a nM | ||
| Citation |  Giri, R; Namballa, HK; Sarker, A; Alberts, I; Harding, WW Synthesis and dopamine receptor pharmacological evaluations on ring C ortho halogenated 1-phenylbenzazepines. Bioorg Med Chem Lett30:0 (2020) [PubMed] Article | ||
| More Info.: | Get all data from this article, Assay Method | ||
| D(1B) dopamine receptor | |||
| Name: | D(1B) dopamine receptor | ||
| Synonyms: | D(5) dopamine receptor | D1beta dopamine receptor | DOPAMINE D5 | DRD1B | DRD1L2 | DRD5 | DRD5_HUMAN | dopamine receptor D5 | ||
| Type: | Protein | ||
| Mol. Mass.: | 52943.41 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | P21918 | ||
| Residue: | 477 | ||
| Sequence: |
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| BDBM50004822 | |||
| n/a | |||
| Name | BDBM50004822 | ||
| Synonyms: | (R)-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol | (R)-7,8-Dihydroxy-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepinium | 1-Phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol | 1-Phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol(SKF38393) | 7,8-Dihydroxy-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepinium(R(+)SKF38393) | CHEMBL1467585 | CHEMBL24077 | R(+)SKF 383931-Phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol | SK&F-383933 | SK-38393 | SK-383933 | SKF 38393 | SKF 38393 (+) | ||
| Type | Small organic molecule | ||
| Emp. Form. | C16H17NO2 | ||
| Mol. Mass. | 255.3117 | ||
| SMILES | Oc1cc2CCNC[C@H](c3ccccc3)c2cc1O | ||
| Structure | 
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