| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide Y receptor type 5 |
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| Ligand | BDBM50103704 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_143985 (CHEMBL750823) |
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| IC50 | >1000±n/a nM |
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| Citation |  Kordik, CP; Luo, C; Zanoni, BC; Dax, SL; McNally, JJ; Lovenberg, TW; Wilson, SJ; Reitz, AB Aminopyrazoles with high affinity for the human neuropeptide Y5 receptor. Bioorg Med Chem Lett11:2283-6 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Neuropeptide Y receptor type 5 |
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| Name: | Neuropeptide Y receptor type 5 |
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| Synonyms: | NPY-Y5 | NPY-Y5 receptor | NPY5-R | NPY5R | NPY5R_HUMAN | NPYR5 | NPYY5 | Neuropeptide Y receptor type 5 | Neuropeptide Y receptor type 5 ( NPY Y5) | Y5 receptor |
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| Type: | Enzyme |
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| Mol. Mass.: | 50746.64 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q15761 |
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| Residue: | 445 |
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| Sequence: | MDLELDEYYNKTLATENNTAATRNSDFPVWDDYKSSVDDLQYFLIGLYTFVSLLGFMGNL
LILMALMKKRNQKTTVNFLIGNLAFSDILVVLFCSPFTLTSVLLDQWMFGKVMCHIMPFL
QCVSVLVSTLILISIAIVRYHMIKHPISNNLTANHGYFLIATVWTLGFAICSPLPVFHSL
VELQETFGSALLSSRYLCVESWPSDSYRIAFTISLLLVQYILPLVCLTVSHTSVCRSISC
GLSNKENRLEENEMINLTLHPSKKSGPQVKLSGSHKWSYSFIKKHRRRYSKKTACVLPAP
ERPSQENHSRILPENFGSVRSQLSSSSKFIPGVPTCFEIKPEENSDVHELRVKRSVTRIK
KRSRSVFYRLTILILVFAVSWMPLHLFHVVTDFNDNLISNRHFKLVYCICHLLGMMSCCL
NPILYGFLNNGIKADLVSLIHCLHM
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| BDBM50103704 |
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| n/a |
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| Name | BDBM50103704 |
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| Synonyms: | CHEMBL73990 | N-[4-(5-Amino-1-p-tolyl-1H-pyrazol-3-yl)-phenyl]-4-methoxy-N-methyl-benzenesulfonamide |
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| Type | Small organic molecule |
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| Emp. Form. | C24H24N4O3S |
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| Mol. Mass. | 448.537 |
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| SMILES | COc1ccc(cc1)S(=O)(=O)N(C)c1ccc(cc1)-c1cc(N)n(n1)-c1ccc(C)cc1 |
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| Structure | 
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