| Reaction Details |
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 | Report a problem with these data |
| Target | Motilin receptor |
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| Ligand | BDBM50108829 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_122666 (CHEMBL732796) |
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| IC50 | 59±n/a nM |
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| Citation |  Haramura, M; Okamachi, A; Tsuzuki, K; Yogo, K; Ikuta, M; Kozono, T; Takanashi, H; Murayama, E Design and synthesis of motilin antagonists derived from the [1-4] fragment of porcine motilin. J Med Chem45:670-5 (2002) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Motilin receptor |
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| Name: | Motilin receptor |
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| Synonyms: | n/a |
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| Type: | n/a |
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| Mol. Mass.: | 43771.25 |
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| Organism: | Oryctolagus cuniculus |
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| Description: | n/a |
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| Residue: | 400 |
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| Sequence: | MGSPWNGSDGPEDAREPPWAALPPCDERRCSPFPLGTLVPVTAVCLGLFAVGVSGNVVTV
LLIGRYRDMRTTTNLYLGSMAVSDLLILLGLPFDLYRLWRSRPWVFGQLLCRLSLYVGEG
CTYASLLHMTALSVERYLAICRPLRARVLVTRRRVRALIAALWAVALLSAGPFFFLVGVE
QDPAVFAAPDRNGTVPLDPSSPAPASPPSGPGAEAAALFSRECRPSRAQLGLLRVMLWVT
TAYFFLPFLCLSILYGLIARQLWRGRGPLRGPAATGRERGHRQTVRVLLVVVLAFIVCWL
PFHVGRIIYINTQDSRMMYFSQYFNIVALQLFYLSASINPILYNLISKKYRAAARRLLRE
SRAGPSGVCGSRGPEQDVAGDTGGDTAGCTETSANTKTAA
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| BDBM50108829 |
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| n/a |
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| Name | BDBM50108829 |
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| Synonyms: | 2-Amino-N-[2-(3-tert-butyl-4-hydroxy-benzyl)-3,8,15-trioxo-1,4,9triaza-cyclopentadec-14-yl]-3-phenyl-propionamide | CHEMBL348744 |
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| Type | Small organic molecule |
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| Emp. Form. | C32H45N5O5 |
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| Mol. Mass. | 579.7302 |
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| SMILES | CC(C)(C)c1cc(CC2NC(=O)C(CCCCNC(=O)CCCNC2=O)NC(=O)C(N)Cc2ccccc2)ccc1O |
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| Structure | 
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