| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Motilin receptor |
|---|
| Ligand | BDBM50108837 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_122666 (CHEMBL732796) |
|---|
| IC50 | 480±n/a nM |
|---|
| Citation |  Haramura, M; Okamachi, A; Tsuzuki, K; Yogo, K; Ikuta, M; Kozono, T; Takanashi, H; Murayama, E Design and synthesis of motilin antagonists derived from the [1-4] fragment of porcine motilin. J Med Chem45:670-5 (2002) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Motilin receptor |
|---|
| Name: | Motilin receptor |
|---|
| Synonyms: | n/a |
|---|
| Type: | n/a |
|---|
| Mol. Mass.: | 43771.25 |
|---|
| Organism: | Oryctolagus cuniculus |
|---|
| Description: | n/a |
|---|
| Residue: | 400 |
|---|
| Sequence: | MGSPWNGSDGPEDAREPPWAALPPCDERRCSPFPLGTLVPVTAVCLGLFAVGVSGNVVTV
LLIGRYRDMRTTTNLYLGSMAVSDLLILLGLPFDLYRLWRSRPWVFGQLLCRLSLYVGEG
CTYASLLHMTALSVERYLAICRPLRARVLVTRRRVRALIAALWAVALLSAGPFFFLVGVE
QDPAVFAAPDRNGTVPLDPSSPAPASPPSGPGAEAAALFSRECRPSRAQLGLLRVMLWVT
TAYFFLPFLCLSILYGLIARQLWRGRGPLRGPAATGRERGHRQTVRVLLVVVLAFIVCWL
PFHVGRIIYINTQDSRMMYFSQYFNIVALQLFYLSASINPILYNLISKKYRAAARRLLRE
SRAGPSGVCGSRGPEQDVAGDTGGDTAGCTETSANTKTAA
|
|
|
|---|
| BDBM50108837 |
|---|
| n/a |
|---|
| Name | BDBM50108837 |
|---|
| Synonyms: | 2-Amino-N-[2-(4-sec-butoxy-benzyl)-3,7,14-trioxo-1,4,8triaza-cyclotetradec-13-yl]-3-phenyl-propionamide | CHEMBL348935 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C31H43N5O5 |
|---|
| Mol. Mass. | 565.7036 |
|---|
| SMILES | CCC(C)Oc1ccc(CC2NC(=O)C(CCCCNC(=O)CCNC2=O)NC(=O)C(N)Cc2ccccc2)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
