| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM50120218 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_147145 |
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| Ki | 141±n/a nM |
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| Citation |  Rinnová, M; Nefzi, A; Houghten, RA Opioid activity of 4-imidazolidinone positional analogues of Leu-Enkephalin. Bioorg Med Chem Lett12:3175-8 (2002) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | D-OR-1 | DOR-1 | Delta opioid receptor | Delta-type opioid receptor (Delta) | OPIATE Delta | OPRD | OPRD1 | OPRD_HUMAN | OPRK1 | opioid receptor, delta 1 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 40382.98 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Competition binding assays were carried out using membrane preparations from transfected HN9.10 cells that constitutively expressed the delta opioid receptor. |
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| Residue: | 372 |
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| Sequence: | MEPAPSAGAELQPPLFANASDAYPSACPSAGANASGPPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTRPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRKPCGRPDPSSFSRAREATARERVTAC
TPSDGPGGGAAA
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| BDBM50120218 |
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| n/a |
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| Name | BDBM50120218 |
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| Synonyms: | (1S,3S)-2-[2-(3-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-acetyl}-5-oxo-imidazolidin-1-yl)-3-phenyl-propionylamino]-4-methyl-pentanoic acid amide | CHEMBL106880 |
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| Type | Small organic molecule |
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| Emp. Form. | C29H38N6O6 |
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| Mol. Mass. | 566.6486 |
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| SMILES | CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)N1CN(CC1=O)C(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(N)=O |
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| Structure | 
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