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TargetSigma intracellular receptor 2
LigandBDBM50562420
Substrate/Competitorn/a
Meas. Tech.ChEMBL_2078427 (CHEMBL4734218)
Ki 130±n/a nM
Citation Kopp, NHoltschulte, CBörgel, FLehmkuhl, KFriedland, KCivenni, GLaurini, ECatapano, CVPricl, SHumpf, HUSchepmann, DWünsch, B Novel ? Eur J Med Chem210:0 (2021) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Sigma intracellular receptor 2
Name:Sigma intracellular receptor 2
Synonyms:S2r | SGMR2_RAT | Sigma intracellular receptor 2 | Sigma-2 receptor | Sigma2 receptor | Tmem97 | Transmembrane protein 97
Type:Protein
Mol. Mass.:20953.88
Organism:Rattus norvegicus (Rat)
Description:Q5U3Y7
Residue:176
Sequence:
MGAVTARRCVEWLLGLYFVSHIPITMFIDLQALLPPELYPQEFSNLLRWYSKEFKDPLMQ
EPPVWFKSFLFCELVFQLPFFPIAAYAFFKGSCRWIRIPAIIYAVHTITTLIPILYTILF
EDFSKAIAFKGQRPENFRERLTLVGVYAPYLIIPLILLLFMLRNPYYKFEEKRKKK
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BDBM50562420
n/a
NameBDBM50562420
Synonyms:CHEMBL4758825
TypeSmall organic molecule
Emp. Form.C21H27N
Mol. Mass.293.4458
SMILESC(C[C@@H]1CCC[C@@H](C1)c1ccccc1)NCc1ccccc1 |r|
Structure
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