| Reaction Details |
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 | Report a problem with these data |
| Target | Atypical chemokine receptor 3 |
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| Ligand | BDBM50567151 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2102410 (CHEMBL4810806) |
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| Ki | 155±n/a nM |
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| Citation |  Aspnes, GE; Menhaji-Klotz, E; Boehm, M; Londregan, AT; Lee, ECY; Limberakis, C; Coffey, SB; Brown, JA; Jones, RM; Hesp, KD Discovery and evaluation of non-basic small molecule modulators of the atypical chemokine receptor CXCR7. Bioorg Med Chem Lett50:0 (2021) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Atypical chemokine receptor 3 |
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| Name: | Atypical chemokine receptor 3 |
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| Synonyms: | ACKR3_MOUSE | Ackr3 | Atypical chemokine receptor 3 | C-X-C chemokine receptor type 7 | CXC-R7 | CXCR-7 | Chemokine orphan receptor 1 | Cmkor1 | Cxcr7 | G-protein coupled receptor RDC1 homolog | RDC-1 | Rdc1 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 41640.48 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_117401 |
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| Residue: | 362 |
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| Sequence: | MDVHLFDYAEPGNYSDINWPCNSSDCIVVDTVQCPTMPNKNVLLYTLSFIYIFIFVIGMI
ANSVVVWVNIQAKTTGYDTHCYILNLAIADLWVVITIPVWVVSLVQHNQWPMGELTCKIT
HLIFSINLFGSIFFLACMSVDRYLSITYFTGTSSYKKKMVRRVVCILVWLLAFFVSLPDT
YYLKTVTSASNNETYCRSFYPEHSIKEWLIGMELVSVILGFAVPFTIIAIFYFLLARAMS
ASGDQEKHSSRKIIFSYVVVFLVCWLPYHFVVLLDIFSILHYIPFTCQLENVLFTALHVT
QCLSLVHCCVNPVLYSFINRNYRYELMKAFIFKYSAKTGLTKLIDASRVSETEYSALEQN
TK
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| BDBM50567151 |
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| n/a |
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| Name | BDBM50567151 |
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| Synonyms: | CHEMBL4848754 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H27N7O2 |
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| Mol. Mass. | 397.4741 |
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| SMILES | [H][C@@]12CN(C[C@]1([H])[C@H]2C(=O)N[C@H]1CCN(C1)c1nccn2ccnc12)C(=O)N(C)CC |r| |
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| Structure | 
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