| Reaction Details |
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 | Report a problem with these data |
| Target | Sigma intracellular receptor 2 |
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| Ligand | BDBM50487259 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2113161 (CHEMBL4822011) |
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| Ki | 7.2±n/a nM |
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| Citation |  Cordone, P; Namballa, HK; Muniz, B; Pal, RK; Gallicchio, E; Harding, WW New tetrahydroisoquinoline-based D Bioorg Med Chem Lett42:0 (2021) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Sigma intracellular receptor 2 |
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| Name: | Sigma intracellular receptor 2 |
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| Synonyms: | MAC30 | Meningioma-associated protein 30 | S2R | SGMR2_HUMAN | Sigma-2 receptor | Sigma2 receptor | TMEM97 | Transmembrane protein 97 |
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| Type: | Protein |
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| Mol. Mass.: | 20857.20 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q5BJF2 |
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| Residue: | 176 |
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| Sequence: | MGAPATRRCVEWLLGLYFLSHIPITLFMDLQAVLPRELYPVEFRNLLKWYAKEFKDPLLQ
EPPAWFKSFLFCELVFQLPFFPIATYAFLKGSCKWIRTPAIIYSVHTMTTLIPILSTFLF
EDFSKASGFKGQRPETLHERLTLVSVYAPYLLIPFILLIFMLRSPYYKYEEKRKKK
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| BDBM50487259 |
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| n/a |
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| Name | BDBM50487259 |
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| Synonyms: | CHEBI:64219 | [3H]NEMONAPRIDE |
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| Type | Small organic molecule |
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| Emp. Form. | C21H26ClN3O2 |
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| Mol. Mass. | 387.903 |
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| SMILES | CNc1cc(OC)c(cc1Cl)C(=O)N[C@@H]1CCN(Cc2ccccc2)[C@@H]1C |r| |
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| Structure | 
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