| Reaction Details |
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 | Report a problem with these data |
| Target | Transient receptor potential cation channel subfamily V member 2 |
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| Ligand | BDBM50285610 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2184546 (CHEMBL5096628) |
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| IC50 | 2200±n/a nM |
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| Citation |  Sampson, PB Phytocannabinoid Pharmacology: Medicinal Properties of J Nat Prod84:142-160 (2021) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Transient receptor potential cation channel subfamily V member 2 |
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| Name: | Transient receptor potential cation channel subfamily V member 2 |
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| Synonyms: | OTRPC2 | Osm-9-like TRP channel 2 | TRPV2 | TRPV2_HUMAN | Transient receptor potential cation channel subfamily V member 2 | VRL | VRL-1 | Vanilloid receptor-like protein 1 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 85972.07 |
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| Organism: | Homo sapiens |
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| Description: | ChEMBL_101052 |
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| Residue: | 764 |
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| Sequence: | MTSPSSSPVFRLETLDGGQEDGSEADRGKLDFGSGLPPMESQFQGEDRKFAPQIRVNLNY
RKGTGASQPDPNRFDRDRLFNAVSRGVPEDLAGLPEYLSKTSKYLTDSEYTEGSTGKTCL
MKAVLNLKDGVNACILPLLQIDRDSGNPQPLVNAQCTDDYYRGHSALHIAIEKRSLQCVK
LLVENGANVHARACGRFFQKGQGTCFYFGELPLSLAACTKQWDVVSYLLENPHQPASLQA
TDSQGNTVLHALVMISDNSAENIALVTSMYDGLLQAGARLCPTVQLEDIRNLQDLTPLKL
AAKEGKIEIFRHILQREFSGLSHLSRKFTEWCYGPVRVSLYDLASVDSCEENSVLEIIAF
HCKSPHRHRMVVLEPLNKLLQAKWDLLIPKFFLNFLCNLIYMFIFTAVAYHQPTLKKQAA
PHLKAEVGNSMLLTGHILILLGGIYLLVGQLWYFWRRHVFIWISFIDSYFEILFLFQALL
TVVSQVLCFLAIEWYLPLLVSALVLGWLNLLYYTRGFQHTGIYSVMIQKVILRDLLRFLL
IYLVFLFGFAVALVSLSQEAWRPEAPTGPNATESVQPMEGQEDEGNGAQYRGILEASLEL
FKFTIGMGELAFQEQLHFRGMVLLLLLAYVLLTYILLLNMLIALMSETVNSVATDSWSIW
KLQKAISVLEMENGYWWCRKKQRAGVMLTVGTKPDGSPDERWCFRVEEVNWASWEQTLPT
LCEDPSGAGVPRTLENPVLASPPKEDEDGASEENYVPVQLLQSN
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| BDBM50285610 |
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| n/a |
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| Name | BDBM50285610 |
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| Synonyms: | CBV | CHEMBL4170268 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H22O2 |
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| Mol. Mass. | 282.3768 |
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| SMILES | CCCc1cc(O)c-2c(OC(C)(C)c3ccc(C)cc-23)c1 |
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| Structure | 
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