| Reaction Details |
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 | Report a problem with these data |
| Target | Transient receptor potential cation channel subfamily V member 3 |
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| Ligand | BDBM50285610 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2184549 (CHEMBL5096631) |
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| IC50 | 1600±n/a nM |
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| Citation |  Sampson, PB Phytocannabinoid Pharmacology: Medicinal Properties of J Nat Prod84:142-160 (2021) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Transient receptor potential cation channel subfamily V member 3 |
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| Name: | Transient receptor potential cation channel subfamily V member 3 |
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| Synonyms: | TRPV3 | TRPV3_HUMAN | Transient receptor potential cation channel subfamily V member 3 (TRPV3) | Vanilloid receptor-like 3 |
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| Type: | Enzyme |
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| Mol. Mass.: | 90635.51 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q8NET8 |
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| Residue: | 790 |
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| Sequence: | MKAHPKEMVPLMGKRVAAPSGNPAILPEKRPAEITPTKKSAHFFLEIEGFEPNPTVAKTS
PPVFSKPMDSNIRQCISGNCDDMDSPQSPQDDVTETPSNPNSPSAQLAKEEQRRKKRRLK
KRIFAAVSEGCVEELVELLVELQELCRRRHDEDVPDFLMHKLTASDTGKTCLMKALLNIN
PNTKEIVRILLAFAEENDILGRFINAEYTEEAYEGQTALNIAIERRQGDIAALLIAAGAD
VNAHAKGAFFNPKYQHEGFYFGETPLALAACTNQPEIVQLLMEHEQTDITSRDSRGNNIL
HALVTVAEDFKTQNDFVKRMYDMILLRSGNWELETTRNNDGLTPLQLAAKMGKAEILKYI
LSREIKEKRLRSLSRKFTDWAYGPVSSSLYDLTNVDTTTDNSVLEITVYNTNIDNRHEML
TLEPLHTLLHMKWKKFAKHMFFLSFCFYFFYNITLTLVSYYRPREEEAIPHPLALTHKMG
WLQLLGRMFVLIWAMCISVKEGIAIFLLRPSDLQSILSDAWFHFVFFIQAVLVILSVFLY
LFAYKEYLACLVLAMALGWANMLYYTRGFQSMGMYSVMIQKVILHDVLKFLFVYIVFLLG
FGVALASLIEKCPKDNKDCSSYGSFSDAVLELFKLTIGLGDLNIQQNSKYPILFLFLLIT
YVILTFVLLLNMLIALMGETVENVSKESERIWRLQRARTILEFEKMLPEWLRSRFRMGEL
CKVAEDDFRLCLRINEVKWTEWKTHVSFLNEDPGPVRRTDFNKIQDSSRNNSKTTLNAFE
EVEEFPETSV
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| BDBM50285610 |
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| n/a |
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| Name | BDBM50285610 |
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| Synonyms: | CBV | CHEMBL4170268 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H22O2 |
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| Mol. Mass. | 282.3768 |
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| SMILES | CCCc1cc(O)c-2c(OC(C)(C)c3ccc(C)cc-23)c1 |
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| Structure | 
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