| Reaction Details |
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 | Report a problem with these data |
| Target | Translocator protein |
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| Ligand | BDBM50229594 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2191878 (CHEMBL5104238) |
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| IC50 | 8.1±n/a nM |
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| Citation |  Barresi, E; Robello, M; Costa, B; Da Pozzo, E; Baglini, E; Salerno, S; Da Settimo, F; Martini, C; Taliani, S An update into the medicinal chemistry of translocator protein (TSPO) ligands. Eur J Med Chem209:0 (2021) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Translocator protein |
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| Name: | Translocator protein |
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| Synonyms: | BZRP | MBR | Mitochondrial benzodiazepine receptor | PBR | PKBS | Peripheral benzodiazepine receptor-related protein | Peripheral-type benzodiazepine receptor | TSPO | TSPO_HUMAN |
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| Type: | Enzyme |
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| Mol. Mass.: | 18834.74 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P30536 |
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| Residue: | 169 |
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| Sequence: | MAPPWVPAMGFTLAPSLGCFVGSRFVHGEGLRWYAGLQKPSWHPPHWVLGPVWGTLYSAM
GYGSYLVWKELGGFTEKAVVPLGLYTGQLALNWAWPPIFFGARQMGWALVDLLLVSGAAA
ATTVAWYQVSPLAARLLYPYLAWLAFTTTLNYCVWRDNHGWRGGRRLPE
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| BDBM50229594 |
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| n/a |
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| Name | BDBM50229594 |
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| Synonyms: | CHEMBL253597 | N-(2-methoxybenzyl)-N-(4-phenoxypyridin-3-yl)acetamide |
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| Type | Small organic molecule |
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| Emp. Form. | C21H20N2O3 |
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| Mol. Mass. | 348.3951 |
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| SMILES | COc1ccccc1CN(C(C)=O)c1cnccc1Oc1ccccc1 |
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| Structure | 
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