| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50594834 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2214487 (CHEMBL5127619) |
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| Ki | 11±n/a nM |
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| Citation |  Smith, MT; Kong, D; Kuo, A; Imam, MZ; Williams, CM Analgesic Opioid Ligand Discovery Based on Nonmorphinan Scaffolds Derived from Natural Sources. J Med Chem65:1612-1661 (2022) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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| BDBM50594834 |
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| n/a |
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| Name | BDBM50594834 |
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| Synonyms: | CHEMBL5178409 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H32N2O5 |
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| Mol. Mass. | 416.5106 |
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| SMILES | [H][C@@]12C[C@@]([H])([C@H](CC)CN1CC[C@@]1(O)C2Nc2cccc(OC)c12)C(=C/OC)\C(=O)OC |r| |
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| Structure | 
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