| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A1 |
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| Ligand | BDBM50260481 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_531569 (CHEMBL990573) |
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| Ki | 4400±n/a nM |
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| Citation |  Raghu Prasad, M; Raghuram Rao, A; Shanthan Rao, P; Rajan, KS; Meena, S; Madhavi, K Synthesis and adenosine receptor binding studies of some novel triazolothienopyrimidines. Eur J Med Chem43:614-20 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A1 |
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| Name: | Adenosine receptor A1 |
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| Synonyms: | AA1R_RAT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptor | Adenosine receptors A1 | Adora1 |
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| Type: | Protein |
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| Mol. Mass.: | 36704.13 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | n/a |
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| Residue: | 326 |
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| Sequence: | MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVT
QRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALIL
FLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCQPKPPIDEDLPEEKAED
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| BDBM50260481 |
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| n/a |
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| Name | BDBM50260481 |
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| Synonyms: | 5-Methyl-8,9,10,11-tetrahydro[1]benzothieno[3,2-e][1,2,4]triazolo[4,3-c]pyrimidine-3(2H)-thione | CHEMBL510505 | cid_714639 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H12N4S2 |
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| Mol. Mass. | 276.38 |
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| SMILES | Cc1nc2sc3CCCCc3c2c2n[nH]c(=S)n12 |
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| Structure | 
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