Reaction Details | |||
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Target | Cholecystokinin receptor type A | ||
Ligand | BDBM50263103 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | ChEMBL_490135 (CHEMBL994440) | ||
IC50 | 1.9±n/a nM | ||
Citation | ![]() | ||
More Info.: | Get all data from this article, Assay Method | ||
Cholecystokinin receptor type A | |||
Name: | Cholecystokinin receptor type A | ||
Synonyms: | CCK-A receptor | CCK-AR | CCK1-R | CCKAR | CCKAR_HUMAN | CCKRA | Cholecystokinin receptor | Cholecystokinin receptor type A | Cholecystokinin-1 Receptor | ||
Type: | G Protein-Coupled Receptor (GPCR) | ||
Mol. Mass.: | 47859.34 | ||
Organism: | Homo sapiens (Human) | ||
Description: | Stable expression of human CCK-1 receptors in HEK 293 cells. | ||
Residue: | 428 | ||
Sequence: |
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BDBM50263103 | |||
n/a | |||
Name | BDBM50263103 | ||
Synonyms: | (2-(2,6-difluorophenyl)-1-(3-ethoxyphenyl)-1H-imidazol-4-yl)(4-(naphthalen-2-yl)piperazin-1-yl)methanone | CHEMBL473457 | ||
Type | Small organic molecule | ||
Emp. Form. | C32H28F2N4O2 | ||
Mol. Mass. | 538.5871 | ||
SMILES | CCOc1cccc(c1)-n1cc(nc1-c1c(F)cccc1F)C(=O)N1CCN(CC1)c1ccc2ccccc2c1 |(-.9,-39.94,;-2.01,-41,;-3.49,-40.57,;-4.61,-41.64,;-6.09,-41.2,;-7.2,-42.28,;-6.84,-43.77,;-5.36,-44.19,;-4.24,-43.13,;-5,-45.69,;-3.49,-46.03,;-3.36,-47.57,;-4.77,-48.17,;-5.79,-47.01,;-7.3,-47.27,;-7.84,-48.71,;-6.85,-49.89,;-9.35,-48.96,;-10.34,-47.77,;-9.8,-46.33,;-8.28,-46.07,;-7.74,-44.63,;-2.03,-48.36,;-2.06,-49.9,;-.69,-47.61,;.64,-48.4,;1.99,-47.66,;2.02,-46.11,;.69,-45.32,;-.66,-46.07,;3.37,-45.37,;3.39,-43.84,;4.73,-43.09,;6.06,-43.88,;7.4,-43.15,;8.71,-43.94,;8.69,-45.48,;7.34,-46.22,;6.02,-45.42,;4.68,-46.17,)| | ||
Structure | ![]() |