| Reaction Details |
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 | Report a problem with these data |
| Target | D(2) dopamine receptor |
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| Ligand | BDBM50220541 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_510243 (CHEMBL1005621) |
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| IC50 | 5±n/a nM |
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| Citation |  Kim, K; Miller, NR; Sulikowski, GA; Lindsley, CW A new multi-gram synthetic route to labeling precursors for the D(2/3) PET agent 18F-fallypride. Bioorg Med Chem Lett18:4467-9 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(2) dopamine receptor |
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| Name: | D(2) dopamine receptor |
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| Synonyms: | D(2) dopamine receptor | DOPAMINE D2 | DOPAMINE D2 Long | DOPAMINE D2 Short | DRD2 | DRD2_HUMAN | Dopamine D2 receptor | Dopamine D2 receptor (D2) | Dopamine D2 receptor (D2R) | Dopamine D2A | Dopamine2-like | d2 |
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| Type: | Cell-surface receptors |
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| Mol. Mass.: | 50647.10 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P14416 |
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| Residue: | 443 |
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| Sequence: | MDPLNLSWYDDDLERQNWSRPFNGSDGKADRPHYNYYATLLTLLIAVIVFGNVLVCMAVS
REKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTA
SILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMISIVWVLSFTISCPLLFGLNNADQN
ECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRRRRKRVNTKRSSRAFRAHLRAPL
KGNCTHPEDMKLCTVIMKSNGSFPVNRRRVEAARRAQELEMEMLSSTSPPERTRYSPIPP
SHHQLTLPDPSHHGLHSTPDSPAKPEKNGHAKDHPKIAKIFEIQTMPNGKTRTSLKTMSR
RKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCDCNIPPVLYSAFTWLGYVNSA
VNPIIYTTFNIEFRKAFLKILHC
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| BDBM50220541 |
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| n/a |
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| Name | BDBM50220541 |
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| Synonyms: | CHEMBL392158 | Fallypride | N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-(3-fluoropropyl)-2,3-dimethoxybenzamide |
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| Type | Small organic molecule |
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| Emp. Form. | C20H29FN2O3 |
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| Mol. Mass. | 364.4543 |
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| SMILES | COc1cc(CCCF)cc(C(=O)NC[C@@H]2CCCN2CC=C)c1OC |r| |
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| Structure | 
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