| Reaction Details |
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 | Report a problem with these data |
| Target | Thromboxane A2 receptor |
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| Ligand | BDBM50281917 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_209595 |
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| Kd | 0.500000±n/a nM |
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| Citation |  Das, J; Hall, SE; Reid, JA; Han, WC; Harris, DN; Goldenberg, H; Michel, IM; Monshizadegan, H; Webb, ML Syntheses of Cyclopentane, Cyclohexene and Olefin Oxazoles as Thromboxane A2/Endoperoxide Receptor Antagonists Bioorg Med Chem Lett3:1267-1270 (1993) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Thromboxane A2 receptor |
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| Name: | Thromboxane A2 receptor |
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| Synonyms: | Prostanoid TP receptor | TA2R_HUMAN | TBXA2R | TXA2-R | Thromboxane | Thromboxane A2 receptor | Thromboxane Beta |
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| Type: | Enyzme |
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| Mol. Mass.: | 37445.28 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21731 |
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| Residue: | 343 |
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| Sequence: | MWPNGSSLGPCFRPTNITLEERRLIASPWFAASFCVVGLASNLLALSVLAGARQGGSHTR
SSFLTFLCGLVLTDFLGLLVTGTIVVSQHAALFEWHAVDPGCRLCRFMGVVMIFFGLSPL
LLGAAMASERYLGITRPFSRPAVASQRRAWATVGLVWAAALALGLLPLLGVGRYTVQYPG
SWCFLTLGAESGDVAFGLLFSMLGGLSVGLSFLLNTVSVATLCHVYHGQEAAQQRPRDSE
VEMMAQLLGIMVVASVCWLPLLVFIAQTVLRNPPAMSPAGQLSRTTEKELLIYLRVATWN
QILDPWVYILFRRAVLRRLQPRLSTRPRSLSLQPQLTQRSGLQ
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| BDBM50281917 |
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| n/a |
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| Name | BDBM50281917 |
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| Synonyms: | 3-(2-{2-[4-(4-Chloro-benzylcarbamoyl)-oxazol-2-yl]-cyclopentylmethyl}-phenyl)-propionic acid | CHEMBL25657 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H27ClN2O4 |
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| Mol. Mass. | 466.957 |
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| SMILES | OC(=O)CCc1ccccc1C[C@@H]1CCC[C@H]1c1nc(co1)C(=O)NCc1ccc(Cl)cc1 |
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| Structure | 
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