| Reaction Details |
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 | Report a problem with these data |
| Target | Plasminogen |
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| Ligand | BDBM50289436 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_222787 |
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| IC50 | 14±n/a nM |
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| Citation |  Tamura, SY; Shamblin, BM; Brunck, TK; Ripka, WC RATIONAL DESIGN, SYNTHESIS, AND SERINE PROTEASE INHIBITORY ACTIVITY OF NOVEL P1-ARGININOYL HETEROCYCLES Bioorg Med Chem Lett7:1359-1364 (1997) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Plasminogen |
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| Name: | Plasminogen |
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| Synonyms: | PLMN_RAT | Plasmin | Plasminogen | Plg |
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| Type: | Protein |
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| Mol. Mass.: | 90541.87 |
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| Organism: | Rattus norvegicus |
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| Description: | Q01177 |
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| Residue: | 812 |
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| Sequence: | MDHKEIILLFLLFLKPGQGDSLDGYVSTQGASLHSLTKKQLAAGSIADCLAKCEGETDFI
CRSFQYHSKEQQCVIMAENSKTSSIIRMRDVILFEKRVYLSECKTGIGKGYRGTMSKTKT
GVTCQKWSDTSPHVPKYSPSTHPSEGLEENYCRNPDNDEQGPWCYTTDPDQRYEYCNIPE
CEEECMYCSGEKYEGKISKTMSGLDCQSWDSQSPHAHGYIPAKFPSKNLKMNYCRNPDGE
PRPWCFTTDPNKRWEYCDIPRCTTPPPPPGPTYQCLKGRGENYRGTVSVTASGKTCQRWS
EQTPHRHNRTPENFPCKNLEENYCRNPDGETAPWCYTTDSQLRWEYCEIPSCGSSVSPDQ
SDSSVLPEQTPVVQECYQGNGKSYRGTSSTTNTGKKCQSWVSMTPHSHSKTPANFPDAGL
EMNYCRNPDNDQRGPWCFTTDPSVRWEYCNLKRCSETGGGVAESAIVPQVPSAPGTSETD
CMYGNGKEYRGKTAVTAAGTPCQEWAAQEPHSHRIFTPQTNPRAGLEKNYCRNPDGDVNG
PWCYTMNPRKLYDYCNIPLCASLSSFECGKPQVEPKKCPGRVVGGCVANPHSWPWQISLR
TRFSGQHFCGGTLISPEWVLTAAHCLEKSSRPEFYKVILGAHEERILGSDVQQIAVTKLV
LEPNDADIALLKLSRPATITDNVIPACLPSPNYVVADRTLCYITGWGETKGTPGAGRLKE
AQLPVIENKVCNRAEYLNNRVKSTELCAGHLAGGIDSCQGDSGGPLVCFEKDKYILQGVT
SWGLGCARPNKPGVYVRVSRYVNWIEREMRND
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| BDBM50289436 |
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| n/a |
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| Name | BDBM50289436 |
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| Synonyms: | (S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-N-[(S)-1-(benzooxazole-2-carbonyl)-4-guanidino-butyl]-3-naphthalen-1-yl-propionamide; TFA | CHEMBL28968 |
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| Type | Small organic molecule |
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| Emp. Form. | C37H39N7O5 |
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| Mol. Mass. | 661.7495 |
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| SMILES | CC(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H](Cc1cccc2ccccc12)C(=O)N[C@@H](CCCNC(N)=N)C(=O)c1nc2ccccc2o1 |
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| Structure | 
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