| Reaction Details |
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 | Report a problem with these data |
| Target | Receptor-type tyrosine-protein phosphatase epsilon |
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| Ligand | BDBM50118762 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_590759 (CHEMBL1050901) |
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| Ki | 45000±n/a nM |
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| Citation |  Vidovic, D; Schürer, SC Knowledge-based characterization of similarity relationships in the human protein-tyrosine phosphatase family for rational inhibitor design. J Med Chem52:6649-59 (2009) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Receptor-type tyrosine-protein phosphatase epsilon |
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| Name: | Receptor-type tyrosine-protein phosphatase epsilon |
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| Synonyms: | PTPRE | PTPRE_HUMAN | Protein-tyrosine phosphatase epsilon | Receptor-type tyrosine-protein phosphatase epsilon | Receptor-type tyrosine-protein phosphatase epsilon (PTPε) |
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| Type: | Protein |
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| Mol. Mass.: | 80646.31 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P23469 |
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| Residue: | 700 |
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| Sequence: | MEPLCPLLLVGFSLPLARALRGNETTADSNETTTTSGPPDPGASQPLLAWLLLPLLLLLL
VLLLAAYFFRFRKQRKAVVSTSDKKMPNGILEEQEQQRVMLLSRSPSGPKKYFPIPVEHL
EEEIRIRSADDCKQFREEFNSLPSGHIQGTFELANKEENREKNRYPNILPNDHSRVILSQ
LDGIPCSDYINASYIDGYKEKNKFIAAQGPKQETVNDFWRMVWEQKSATIVMLTNLKERK
EEKCHQYWPDQGCWTYGNIRVCVEDCVVLVDYTIRKFCIQPQLPDGCKAPRLVSQLHFTS
WPDFGVPFTPIGMLKFLKKVKTLNPVHAGPIVVHCSAGVGRTGTFIVIDAMMAMMHAEQK
VDVFEFVSRIRNQRPQMVQTDMQYTFIYQALLEYYLYGDTELDVSSLEKHLQTMHGTTTH
FDKIGLEEEFRKLTNVRIMKENMRTGNLPANMKKARVIQIIPYDFNRVILSMKRGQEYTD
YINASFIDGYRQKDYFIATQGPLAHTVEDFWRMIWEWKSHTIVMLTEVQEREQDKCYQYW
PTEGSVTHGEITIEIKNDTLSEAISIRDFLVTLNQPQARQEEQVRVVRQFHFHGWPEIGI
PAEGKGMIDLIAAVQKQQQQTGNHPITVHCSAGAGRTGTFIALSNILERVKAEGLLDVFQ
AVKSLRLQRPHMVQTLEQYEFCYKVVQDFIDIFSDYANFK
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| BDBM50118762 |
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| n/a |
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| Name | BDBM50118762 |
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| Synonyms: | 2-(Oxalyl-amino)-4,5,6,7-tetrahydro-benzo[b]thiophene-3-carboxylic acid | 2-(carboxyformamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylic acid | 2-oxalylamino-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylic acid | CHEMBL138152 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H11NO5S |
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| Mol. Mass. | 269.274 |
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| SMILES | OC(=O)C(=O)Nc1sc2CCCCc2c1C(O)=O |
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| Structure | 
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