| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 3 |
|---|
| Ligand | BDBM50227099 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_621604 (CHEMBL1113036) |
|---|
| Ki | >10000±n/a nM |
|---|
| Citation |  Martin, RE; Mohr, P; Maerki, HP; Guba, W; Kuratli, C; Gavelle, O; Binggeli, A; Bendels, S; Alvarez-Sánchez, R; Alker, A; Polonchuk, L; Christ, AD Benzoxazole piperidines as selective and potent somatostatin receptor subtype 5 antagonists. Bioorg Med Chem Lett19:6106-13 (2009) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Somatostatin receptor type 3 |
|---|
| Name: | Somatostatin receptor type 3 |
|---|
| Synonyms: | SOMATOSTATIN SST3 | SS-3-R | SS3-R | SS3R | SSR-28 | SSR3_HUMAN | SSTR3 | Somatostatin receptor type 3 (SSTR3) |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 45855.97 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P32745 |
|---|
| Residue: | 418 |
|---|
| Sequence: | MDMLHPSSVSTTSEPENASSAWPPDATLGNVSAGPSPAGLAVSGVLIPLVYLVVCVVGLL
GNSLVIYVVLRHTASPSVTNVYILNLALADELFMLGLPFLAAQNALSYWPFGSLMCRLVM
AVDGINQFTSIFCLTVMSVDRYLAVVHPTRSARWRTAPVARTVSAAVWVASAVVVLPVVV
FSGVPRGMSTCHMQWPEPAAAWRAGFIIYTAALGFFGPLLVICLCYLLIVVKVRSAGRRV
WAPSCQRRRRSERRVTRMVVAVVALFVLCWMPFYVLNIVNVVCPLPEEPAFFGLYFLVVA
LPYANSCANPILYGFLSYRFKQGFRRVLLRPSRRVRSQEPTVGPPEKTEEEDEEEEDGEE
SREGGKGKEMNGRVSQITQPGTSGQERPPSRVASKEQQLLPQEASTGEKSSTMRISYL
|
|
|
|---|
| BDBM50227099 |
|---|
| n/a |
|---|
| Name | BDBM50227099 |
|---|
| Synonyms: | 2-(1-(4-amino-3,5-diethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-sulfonamide | CHEMBL236788 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C23H31N5O5S |
|---|
| Mol. Mass. | 489.588 |
|---|
| SMILES | CCOc1cc(CN2CCC(CC2)Nc2nc3cc(ccc3o2)S(N)(=O)=O)cc(OCC)c1N |
|---|
| Structure | 
|
|---|
Search and Browse
