| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide Y receptor type 5 |
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| Ligand | BDBM50355852 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_775165 (CHEMBL1912470) |
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| Ki | 5.4±n/a nM |
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| Citation |  Packiarajan, M; Coate, H; Desai, M; Jimenez, HN; Reinhard, EJ; Jubian, VJ; Marzabadi, MR; Chandrasena, G; Wolinski, TC; Walker, MW; Andersen, K 5-(2'-Pyridyl)-2-aminothiazoles: alkyl amino sulfonamides and sulfamides as potent NPY(5) antagonists. Bioorg Med Chem Lett21:6500-4 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Neuropeptide Y receptor type 5 |
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| Name: | Neuropeptide Y receptor type 5 |
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| Synonyms: | NPY-Y5 | NPY5R_RAT | Neuropeptide Y receptor type 5 | Npy5r | Npyr5 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 50435.58 |
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| Organism: | Rat 6B |
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| Description: | NPY-Y5 NPY5R Rat 6B::Q63634 |
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| Residue: | 445 |
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| Sequence: | MEFKLEEHFNKTFVTENNTAAARNAAFPAWEDYRGSVDDLQYFLIGLYTFVSLLGFMGNL
LILMAVMKKRNQKTTVNFLIGNLAFSDILVVLFCSPFTLTSVLLDQWMFGKAMCHIMPFL
QCVSVLVSTLILISIAIVRYHMIKHPISNNLTANHGYFLIATVWTLGFAICSPLPVFHSL
VELKETFGSALLSSKYLCVESWPSDSYRIAFTISLLLVQYILPLVCLTVSHTSVCRSISC
GLSHKENRLEENEMINLTLQPSKKSRNQAKTPSTQKWSYSFIRKHRRRYSKKTACVLPAP
AGPSQGKHLAVPENPASVRSQLSPSSKVIPGVPICFEVKPEESSDAHEMRVKRSITRIKK
RSRSVFYRLTILILVFAVSWMPLHVFHVVTDFNDNLISNRHFKLVYCICHLLGMMSCCLN
PILYGFLNNGIKADLRALIHCLHMS
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| BDBM50355852 |
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| n/a |
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| Name | BDBM50355852 |
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| Synonyms: | CHEMBL1909725 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H23N5O2S2 |
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| Mol. Mass. | 369.505 |
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| SMILES | CN(C)S(=O)(=O)NCCCCCNc1nc(cs1)-c1ccccn1 |
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| Structure | 
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