| Reaction Details |
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 | Report a problem with these data |
| Target | Dipeptidyl peptidase 1 |
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| Ligand | BDBM50147186 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_44964 |
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| Ki | 514000±n/a nM |
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| Citation |  Mucha, A; Pawel, M; Hurek, J; Kafarski, P Synthesis and activity of phosphinic tripeptide inhibitors of cathepsin C. Bioorg Med Chem Lett14:3113-6 (2004) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Dipeptidyl peptidase 1 |
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| Name: | Dipeptidyl peptidase 1 |
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| Synonyms: | CATC_MOUSE | Ctsc | Dipeptidyl peptidase I |
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| Type: | PROTEIN |
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| Mol. Mass.: | 52379.83 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_44964 |
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| Residue: | 462 |
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| Sequence: | MGPWTHSLRAVLLLVLLGVCTVRSDTPANCTYPDLLGTWVFQVGPRSSRSDINCSVMEAT
EEKVVVHLKKLDTAYDELGNSGHFTLIYNQGFEIVLNDYKWFAFFKYEVRGHTAISYCHE
TMTGWVHDVLGRNWACFVGKKVESHIEKVNMNAAHLGGLQERYSERLYTHNHNFVKAINT
VQKSWTATAYKEYEKMSLRDLIRRSGHSQRIPRPKPAPMTDEIQQQILNLPESWDWRNVQ
GVNYVSPVRNQESCGSCYSFASMGMLEARIRILTNNSQTPILSPQEVVSCSPYAQGCDGG
FPYLIAGKYAQDFGVVEESCFPYTAKDSPCKPRENCLRYYSSDYYYVGGFYGGCNEALMK
LELVKHGPMAVAFEVHDDFLHYHSGIYHHTGLSDPFNPFELTNHAVLLVGYGRDPVTGIE
YWIIKNSWGSNWGESGYFRIRRGTDECAIESIAVAAIPIPKL
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| BDBM50147186 |
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| n/a |
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| Name | BDBM50147186 |
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| Synonyms: | 3-{[1-(2-Amino-acetylamino)-2-phenyl-ethyl]-hydroxy-phosphinoyl}-propionic acid methyl ester; hydrochloride | CHEMBL552867 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H21N2O5P |
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| Mol. Mass. | 328.3007 |
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| SMILES | COC(=O)CCP(O)(=O)C(Cc1ccccc1)NC(=O)CN |
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| Structure | 
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