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TargetSigma non-opioid intracellular receptor 1
LigandBDBM50039200
Substrate/Competitorn/a
Meas. Tech.ChEMBL_201102 (CHEMBL807583)
Ki 2±n/a nM
Citation Calderon, SNIzenwasser, SHeller, BGutkind, JSMattson, MVSu, TPNewman, AH Novel 1-phenylcycloalkanecarboxylic acid derivatives are potent and selective sigma 1 ligands. J Med Chem37:2285-91 (1994) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Sigma non-opioid intracellular receptor 1
Name:Sigma non-opioid intracellular receptor 1
Synonyms:Opioid receptor | Oprs1 | SGMR1_RAT | Sigma | Sigma non-opioid intracellular receptor 1 | Sigma opioid receptor | Sigma-1 | Sigmar1
Type:Enzyme Catalytic Domain
Mol. Mass.:25266.54
Organism:RAT
Description:Q9R0C9
Residue:223
Sequence:
MPWAVGRRWAWITLFLTIVAVLIQAVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSHGHSGRY
WAEISDTIISGTFHQWREGTTKSEVYYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALSDTIFSTQDFLTLFYTLRAYARGLRLELTTYLFGQDP
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  Blast E-value cutoff:
BDBM50039200
n/a
NameBDBM50039200
Synonyms:(4-Phenyl-butyl)-(5-phenyl-pentyl)-amine | CHEMBL20153
TypeSmall organic molecule
Emp. Form.C21H29N
Mol. Mass.295.4617
SMILESC(CCNCCCCc1ccccc1)CCc1ccccc1
Structure
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