| Reaction Details |
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 | Report a problem with these data |
| Target | Galanin receptor type 3 |
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| Ligand | BDBM50273369 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_561971 (CHEMBL1010034) |
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| Kd | 40±n/a nM |
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| Citation |  Bulaj, G; Green, BR; Lee, HK; Robertson, CR; White, K; Zhang, L; Sochanska, M; Flynn, SP; Scholl, EA; Pruess, TH; Smith, MD; White, HS Design, synthesis, and characterization of high-affinity, systemically-active galanin analogues with potent anticonvulsant activities. J Med Chem51:8038-47 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Galanin receptor type 3 |
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| Name: | Galanin receptor type 3 |
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| Synonyms: | GALNR3 | GALR3 | GALR3_HUMAN | Galanin R3 | Galanin receptor 3 | Galanin receptor type 3 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 39599.97 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Galanin R3 GALR3 HUMAN::O60755 |
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| Residue: | 368 |
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| Sequence: | MADAQNISLDSPGSVGAVAVPVVFALIFLLGTVGNGLVLAVLLQPGPSAWQEPGSTTDLF
ILNLAVADLCFILCCVPFQATIYTLDAWLFGALVCKAVHLLIYLTMYASSFTLAAVSVDR
YLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDAR
RRALDVATFAAGYLLPVAVVSLAYGRTLRFLWAAVGPAGAAAAEARRRATGRAGRAMLAV
AALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYALASRHFRA
RFRRLWPCGRRRRHRARRALRRVRPASSGPPGCPGDARPSGRLLAGGGQGPEPREGPVHG
GEAARGPE
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| BDBM50273369 |
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| n/a |
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| Name | BDBM50273369 |
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| Synonyms: | CHEMBL526003 | GWTLNSAGYLLGPQQFFGLM-CONH2 | Galanin (1-13)-SP-(5-11) | galantide |
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| Type | Small organic molecule |
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| Emp. Form. | C104H151N25O26S |
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| Mol. Mass. | 2199.529 |
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| SMILES | CSCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(N)=O |r| |
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| Structure | 
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