| Reaction Details |
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 | Report a problem with these data |
| Target | D(3) dopamine receptor |
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| Ligand | BDBM50039791 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_860682 (CHEMBL2167999) |
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| Ki | 23.9±n/a nM |
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| Citation |  Newman, AH; Beuming, T; Banala, AK; Donthamsetti, P; Pongetti, K; LaBounty, A; Levy, B; Cao, J; Michino, M; Luedtke, RR; Javitch, JA; Shi, L Molecular determinants of selectivity and efficacy at the dopamine D3 receptor. J Med Chem55:6689-99 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(3) dopamine receptor |
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| Name: | D(3) dopamine receptor |
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| Synonyms: | DOPAMINE D3 | DRD3 | DRD3_HUMAN | Dopamine D3 receptor | Dopamine D3 receptor (D3) | Dopamine D3 receptor (D3R) | Dopamine receptor | Dopamine receptor (D3) | Dopamine receptor D3 |
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| Type: | n/a |
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| Mol. Mass.: | 44243.43 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 400 |
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| Sequence: | MASLSQLSSHLNYTCGAENSTGASQARPHAYYALSYCALILAIVFGNGLVCMAVLKERAL
QTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRICCDVFVTLDVMMCTASILN
LCAISIDRYTAVVMPVHYQHGTGQSSCRRVALMITAVWVLAFAVSCPLLFGFNTTGDPTV
CSISNPDFVIYSSVVSFYLPFGVTVLVYARIYVVLKQRRRKRILTRQNSQCNSVRPGFPQ
QTLSPDPAHLELKRYYSICQDTALGGPGFQERGGELKREEKTRNSLSPTIAPKLSLEVRK
LSNGRLSTSLKLGPLQPRGVPLREKKATQMVAIVLGAFIVCWLPFFLTHVLNTHCQTCHV
SPELYSATTWLGYVNSALNPVIYTTFNIEFRKAFLKILSC
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| BDBM50039791 |
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| n/a |
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| Name | BDBM50039791 |
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| Synonyms: | 1-Butyl-4-(2-methoxy-phenyl)-piperazine | CHEMBL26789 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H24N2O |
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| Mol. Mass. | 248.3639 |
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| SMILES | CCCCN1CCN(CC1)c1ccccc1OC |
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| Structure | 
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