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TargetBcl-2-related protein A1
LigandBDBM50397584
Substrate/Competitorn/a
Meas. Tech.ChEMBL_862260 (CHEMBL2173037)
EC50 17800±n/a nM
Citation Saugues, EDebaud, ALAnizon, FBonnefoy, NMoreau, P Synthesis and biological activities of polyquinoline derivatives: new Bcl-2 family protein modulators. Eur J Med Chem57:112-25 (2012) [PubMed]  Article
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Bcl-2-related protein A1
Name:Bcl-2-related protein A1
Synonyms:B2LA1_HUMAN | BCL2A1 | BCL2L5 | BFL1 | Bcl-2-like protein 5 | GRS | HBPA1 | Hemopoietic-specific early response protein | Protein BFL-1 | Protein GRS
Type:Apoptosis regulator protein
Mol. Mass.:20130.01
Organism:Homo sapiens (Human)
Description:n/a
Residue:175
Sequence:
MTDCEFGYIYRLAQDYLQCVLQIPQPGSGPSKTSRVLQNVAFSVQKEVEKNLKSCLDNVN
VVSVDTARTLFNQVMEKEFEDGIINWGRIVTIFAFEGILIKKLLRQQIAPDVDTYKEISY
FVAEFIMNNTGEWIRQNGGWENGFVKKFEPKSGWMTFLEVTGKICEMLSLLKQYC
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BDBM50397584
n/a
NameBDBM50397584
Synonyms:CHEMBL2171506
TypeSmall organic molecule
Emp. Form.C28H31N3O2
Mol. Mass.441.5646
SMILESCCCOc1nc2ccccc2cc1-c1cc(C(C)C)c2ccc(nc2c1)N1CCOCC1
Structure
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