| Reaction Details |
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 | Report a problem with these data |
| Target | RYamide receptor |
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| Ligand | BDBM50192742 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1613599 (CHEMBL3855399) |
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| EC50 | 20900±n/a nM |
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| Citation |  Yoon, YK; Kim, JH; Kim, JH; Kwon, JY; Kim, YC; Kim, YJ; Park, ZY Pyrazolodiazepine derivatives with agonist activity toward Drosophila RYamide receptor. Bioorg Med Chem Lett26:5116-5118 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| RYamide receptor |
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| Name: | RYamide receptor |
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| Synonyms: | NPY-R | NepYr | Neuropeptide Y-like receptor | RYAR_DROME | RYa-R | RYamide receptor | Synonyms=NepYr |
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| Type: | PROTEIN |
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| Mol. Mass.: | 53538.04 |
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| Organism: | Drosophila melanogaster |
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| Description: | ChEMBL_116973 |
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| Residue: | 464 |
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| Sequence: | MEHHNSHLLPGGSEKMYYIAHQQPMLRNEDDNYQEGYFIRPDPASLIYNTTALPADDEGS
NYGYGSTTTLSGLQFETYNITVMMNFSCDDYDLLSEDMWSSAYFKIIVYMLYIPIFIFAL
IGNGTVCYIVYSTPRMRTVTNYFIASLAIGDILMSFFCVPSSFISLFILNYWPFGLALCH
FVNYSQAVSVLVSAYTLVAISIDRYIAIMWPLKPRITKRYATFIIAGVWFIALATALPIP
IVSGLDIPMSPWHTKCEKYICREMWPSRTQEYYYTLSLFALQFVVPLGVLIFTYARITIR
VWAKRPPGEAETNRDQRMARSKRKMVKMMLTVVIVFTCCWLPFNILQLLLNDEEFAHWDP
LPYVWFAFHWLAMSHCCYNPIIYCYMNARFRSGFVQLMHRMPGLRRWCCLRSVGDRMNAT
SGTGPALPLNRMNTSTTYISARRKPRATSLRANPLSCGETSPLR
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| BDBM50192742 |
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| n/a |
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| Name | BDBM50192742 |
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| Synonyms: | CHEMBL3982272 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H39N7OS |
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| Mol. Mass. | 437.646 |
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| SMILES | CC(C)CN1C[C@@H](CCCCN)N=C(SCCC(=O)NN)c2nn(CC(C)C)cc12 |r,t:12| |
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| Structure | 
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