| Reaction Details |
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 | Report a problem with these data |
| Target | Free fatty acid receptor 4 |
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| Ligand | BDBM50196402 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1618417 (CHEMBL3860586) |
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| EC50 | 138±n/a nM |
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| Citation |  Azevedo, CM; Watterson, KR; Wargent, ET; Hansen, SV; Hudson, BD; Kepczynska, MA; Dunlop, J; Shimpukade, B; Christiansen, E; Milligan, G; Stocker, CJ; Ulven, T Non-Acidic Free Fatty Acid Receptor 4 Agonists with Antidiabetic Activity. J Med Chem59:8868-8878 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Free fatty acid receptor 4 |
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| Name: | Free fatty acid receptor 4 |
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| Synonyms: | FFAR4 | FFAR4_HUMAN | G-protein coupled receptor 120 | G-protein coupled receptor 129 | G-protein coupled receptor GT01 | G-protein coupled receptor PGR4 | GPR120 | GPR129 | O3FAR1 | Omega-3 fatty acid receptor 1 | PGR4 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 42256.91 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1508994 |
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| Residue: | 377 |
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| Sequence: | MSPECARAAGDAPLRSLEQANRTRFPFFSDVKGDHRLVLAAVETTVLVLIFAVSLLGNVC
ALVLVARRRRRGATACLVLNLFCADLLFISAIPLVLAVRWTEAWLLGPVACHLLFYVMTL
SGSVTILTLAAVSLERMVCIVHLQRGVRGPGRRARAVLLALIWGYSAVAALPLCVFFRVV
PQRLPGADQEISICTLIWPTIPGEISWDVSFVTLNFLVPGLVIVISYSKILQTSEHLLDA
RAVVTHSEITKASRKRLTVSLAYSESHQIRVSQQDFRLFRTLFLLMVSFFIMWSPIIITI
LLILIQNFKQDLVIWPSLFFWVVAFTFANSALNPILYNMTLCRNEWKKIFCCFWFPEKGA
ILTDTSVKRNDLSIISG
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| BDBM50196402 |
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| n/a |
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| Name | BDBM50196402 |
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| Synonyms: | CHEMBL3910333 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H13ClN2O3S |
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| Mol. Mass. | 372.825 |
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| SMILES | Clc1cc(Oc2ccccn2)cc(c1)N1Cc2ccccc2S1(=O)=O |
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| Structure | 
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