| Reaction Details |
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 | Report a problem with these data |
| Target | Probable G-protein coupled receptor 34 |
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| Ligand | BDBM50238933 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1664557 (CHEMBL4014238) |
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| EC50 | 300±n/a nM |
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| Citation |  Sayama, M; Sayama, M; Sayama, M; Inoue, A; Inoue, A; Inoue, A; Nakamura, S; Nakamura, S; Nakamura, S; Jung, S; Jung, S; Jung, S; Ikubo, M; Ikubo, M; Ikubo, M; Otani, Y; Otani, Y; Otani, Y; Uwamizu, A; Uwamizu, A; Uwamizu, A; Kishi, T; Kishi, T; Kishi, T; Makide, K; Makide, K; Makide, K; Aoki, J; Aoki, J; Aoki, J; Hirokawa, T; Hirokawa, T; Hirokawa, T; Ohwada, T; Ohwada, T; Ohwada, T Probing the Hydrophobic Binding Pocket of G-Protein-Coupled Lysophosphatidylserine Receptor GPR34/LPS J Med Chem60:6384-6399 (2017) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Probable G-protein coupled receptor 34 |
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| Name: | Probable G-protein coupled receptor 34 |
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| Synonyms: | GPR34 | GPR34_HUMAN | Probable G-protein coupled receptor 34 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 43892.32 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_109761 |
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| Residue: | 381 |
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| Sequence: | MRSHTITMTTTSVSSWPYSSHRMRFITNHSDQPPQNFSATPNVTTCPMDEKLLSTVLTTS
YSVIFIVGLVGNIIALYVFLGIHRKRNSIQIYLLNVAIADLLLIFCLPFRIMYHINQNKW
TLGVILCKVVGTLFYMNMYISIILLGFISLDRYIKINRSIQQRKAITTKQSIYVCCIVWM
LALGGFLTMIILTLKKGGHNSTMCFHYRDKHNAKGEAIFNFILVVMFWLIFLLIILSYIK
IGKNLLRISKRRSKFPNSGKYATTARNSFIVLIIFTICFVPYHAFRFIYISSQLNVSSCY
WKEIVHKTNEIMLVLSSFNSCLDPVMYFLMSSNIRKIMCQLLFRRFQGEPSRSESTSEFK
PGYSLHDTSVAVKIQSSSKST
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| BDBM50238933 |
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| n/a |
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| Name | BDBM50238933 |
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| Synonyms: | CHEMBL4089962 |
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| Type | Small organic molecule |
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| Emp. Form. | C32H40NO10P |
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| Mol. Mass. | 629.6345 |
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| SMILES | CC(C)(C)c1ccc(Oc2cccc(COc3ccccc3CCC(=O)OCCCOP(O)(=O)OC[C@H](N)C(O)=O)c2)cc1 |r| |
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| Structure | 
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