| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Kappa-type opioid receptor |
|---|
| Ligand | BDBM86258 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 113±n/a nM |
|---|
| Comments | PDSP_1250 |
|---|
| Citation |  Spetea, M; Tóth, F; Schütz, J; Otvös, F; Tóth, G; Benyhe, S; Borsodi, A; Schmidhammer, H Binding characteristics of [3H]14-methoxymetopon, a high affinity mu-opioid receptor agonist. Eur J Neurosci18:290-5 (2003) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Kappa-type opioid receptor |
|---|
| Name: | Kappa-type opioid receptor |
|---|
| Synonyms: | KOR-1 | Kappa Opioid Receptor | OPIATE Kappa | OPRK_RAT | Opioid receptor | Oprk1 | Ror-d |
|---|
| Type: | G Protein-Coupled Receptor (GPCR) |
|---|
| Mol. Mass.: | 42692.90 |
|---|
| Organism: | Rattus norvegicus (rat) |
|---|
| Description: | P34975 |
|---|
| Residue: | 380 |
|---|
| Sequence: | MESPIQIFRGEPGPTCAPSACLLPNSSSWFPNWAESDSNGSVGSEDQQLEPAHISPAIPV
IITAVYSVVFVVGLVGNSLVMFVIIRYTKMKTATNIYIFNLALADALVTTTMPFQSAVYL
MNSWPFGDVLCKIVISIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPLKAKIINI
CIWLLASSVGISAIVLGGTKVREDVDVIECSLQFPDDEYSWWDLFMKICVFVFAFVIPVL
IIIVCYTLMILRLKSVRLLSGSREKDRNLRRITKLVLVVVAVFIICWTPIHIFILVEALG
STSHSTAVLSSYYFCIALGYTNSSLNPVLYAFLDENFKRCFRDFCFPIKMRMERQSTNRV
RNTVQDPASMRDVGGMNKPV
|
|
|
|---|
| BDBM86258 |
|---|
| n/a |
|---|
| Name | BDBM86258 |
|---|
| Synonyms: | CAS_23552-18-3 | Morphine | NSC_5980 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C17H19NO3 |
|---|
| Mol. Mass. | 285.3377 |
|---|
| SMILES | CN1CCC23C4Oc5c2c(CC1C3C=CC4O)ccc5O |c:16,TLB:13:12:1.2.3:10.9.8| |
|---|
| Structure | 
|
|---|
Search and Browse
