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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Fibroblast growth factor receptor 3 | ||
| Ligand | BDBM102507 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Kinase Assay | ||
| IC50 | >10000±0.0 nM | ||
| Citation |  Furet, P; Graus Porta, D; Guagnano, V Quinoxaline carboxamide derivatives as protein tyrosine kinase inhibitors US Patent US8536175 Publication Date 9/17/2013 | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Fibroblast growth factor receptor 3 | |||
| Name: | Fibroblast growth factor receptor 3 | ||
| Synonyms: | CD_antigen: CD333 | FGFR-3 | FGFR3 | FGFR3_HUMAN | Fibroblast growth factor receptor | Fibroblast growth factor receptor 3 (FGFR3) | JTK4 | ||
| Type: | Protein | ||
| Mol. Mass.: | 87699.57 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | P22607 | ||
| Residue: | 806 | ||
| Sequence: |
| ||
| BDBM102507 | |||
| n/a | |||
| Name | BDBM102507 | ||
| Synonyms: | US8536175, 17 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C19H14Cl2N6O3 | ||
| Mol. Mass. | 445.259 | ||
| SMILES | COc1cc(OC)c(Cl)c(c1Cl)-c1ccc(C(=O)Nc2nnc[nH]2)c2nccnc12 |(5.42,4,;6.19,2.67,;5.42,1.33,;6.19,,;5.42,-1.33,;6.19,-2.67,;7.73,-2.67,;3.88,-1.33,;3.11,-2.67,;3.11,,;3.88,1.33,;3.11,2.67,;1.57,,;.8,1.33,;-.74,1.33,;-1.51,,;-3.05,,;-3.82,1.33,;-3.82,-1.33,;-5.36,-1.33,;-6.27,-2.58,;-7.73,-2.1,;-7.73,-.56,;-6.27,-.09,;-.74,-1.33,;-1.51,-2.67,;-.74,-4,;.8,-4,;1.57,-2.67,;.8,-1.33,)| | ||
| Structure | 
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