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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Neuropeptide Y receptor type 5 | ||
| Ligand | BDBM118178 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Binding Assay | ||
| pH | 7.4±n/a | ||
| Temperature | 298.15±n/a K | ||
| IC50 | 0.65±n/a nM | ||
| Comments | extracted | ||
| Citation |  Yoshida, H; Tonogaki, K; Sakagami, M; Takaya, K Cyclohexane derivative having NPY Y5 receptor antagonism US Patent US8653125 Publication Date 2/18/2014 | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Neuropeptide Y receptor type 5 | |||
| Name: | Neuropeptide Y receptor type 5 | ||
| Synonyms: | NPY-Y5 | NPY5R_MOUSE | Neuropeptide Y receptor Y5 | Neuropeptide Y receptor type 5 (NPY Y5) | Npy5 | Npy5r | ||
| Type: | Enzyme | ||
| Mol. Mass.: | 52807.91 | ||
| Organism: | Mus musculus (Mouse) | ||
| Description: | O70342 | ||
| Residue: | 466 | ||
| Sequence: |
| ||
| BDBM118178 | |||
| n/a | |||
| Name | BDBM118178 | ||
| Synonyms: | US8653125, Ia-35 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C23H23N3O3 | ||
| Mol. Mass. | 389.447 | ||
| SMILES | O=C(Nc1ccc(cc1)-c1ccccc1)[C@@H]1CC[C@@H](CC1)NC(=O)c1ccon1 |r,wU:18.23,15.16,(.52,-1.78,;.52,-.24,;1.85,.53,;3.19,-.24,;3.19,-1.78,;4.52,-2.55,;5.85,-1.78,;5.85,-.24,;4.52,.53,;7.19,-2.55,;7.19,-4.09,;8.52,-4.86,;9.85,-4.09,;9.85,-2.55,;8.52,-1.78,;-.82,.53,;-.82,2.07,;-2.15,2.84,;-3.48,2.07,;-3.48,.53,;-2.15,-.24,;-4.82,2.84,;-6.15,2.07,;-6.15,.53,;-7.48,2.84,;-8.95,2.37,;-9.85,3.61,;-8.95,4.86,;-7.48,4.38,)| | ||
| Structure | 
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