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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Neuropeptide Y receptor type 5 | ||
| Ligand | BDBM118183 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Binding Assay | ||
| pH | 7.4±n/a | ||
| Temperature | 298.15±n/a K | ||
| IC50 | 1.5±n/a nM | ||
| Comments | extracted | ||
| Citation |  Yoshida, H; Tonogaki, K; Sakagami, M; Takaya, K Cyclohexane derivative having NPY Y5 receptor antagonism US Patent US8653125 Publication Date 2/18/2014 | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Neuropeptide Y receptor type 5 | |||
| Name: | Neuropeptide Y receptor type 5 | ||
| Synonyms: | NPY-Y5 | NPY5R_MOUSE | Neuropeptide Y receptor Y5 | Neuropeptide Y receptor type 5 (NPY Y5) | Npy5 | Npy5r | ||
| Type: | Enzyme | ||
| Mol. Mass.: | 52807.91 | ||
| Organism: | Mus musculus (Mouse) | ||
| Description: | O70342 | ||
| Residue: | 466 | ||
| Sequence: |
| ||
| BDBM118183 | |||
| n/a | |||
| Name | BDBM118183 | ||
| Synonyms: | US8653125, Ib-4 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C22H25FN4O3 | ||
| Mol. Mass. | 412.4573 | ||
| SMILES | CC(C)n1c2ccc(NC(=O)[C@@H]3CC[C@@H](CC3)Nc3cccc(F)n3)cc2oc1=O |r,wU:14.17,11.10,(6.82,-3.84,;7.91,-2.75,;9.4,-3.15,;7.51,-1.26,;6.05,-.78,;4.71,-1.55,;3.38,-.78,;3.38,.76,;2.05,1.53,;.71,.76,;.71,-.78,;-.62,1.53,;-.62,3.07,;-1.95,3.84,;-3.29,3.07,;-3.29,1.53,;-1.95,.76,;-4.62,3.84,;-5.96,3.07,;-5.96,1.53,;-7.29,.76,;-8.62,1.53,;-8.62,3.07,;-9.96,3.84,;-7.29,3.84,;4.71,1.53,;6.05,.76,;7.51,1.23,;8.42,-.01,;9.96,-.01,)| | ||
| Structure | 
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