Reaction Details | |||
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Report a problem with these data | |||
Target | Neuropeptide Y receptor type 5 | ||
Ligand | BDBM118191 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | Binding Assay | ||
pH | 7.4±n/a | ||
Temperature | 298.15±n/a K | ||
IC50 | 0.69±n/a nM | ||
Comments | extracted | ||
Citation | Yoshida, H; Tonogaki, K; Sakagami, M; Takaya, K Cyclohexane derivative having NPY Y5 receptor antagonism US Patent US8653125 Publication Date 2/18/2014 | ||
More Info.: | Get all data from this article, Assay Method | ||
Neuropeptide Y receptor type 5 | |||
Name: | Neuropeptide Y receptor type 5 | ||
Synonyms: | NPY-Y5 | NPY5R_MOUSE | Neuropeptide Y receptor Y5 | Neuropeptide Y receptor type 5 (NPY Y5) | Npy5 | Npy5r | ||
Type: | Enzyme | ||
Mol. Mass.: | 52807.91 | ||
Organism: | Mus musculus (Mouse) | ||
Description: | O70342 | ||
Residue: | 466 | ||
Sequence: |
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BDBM118191 | |||
n/a | |||
Name | BDBM118191 | ||
Synonyms: | US8653125, Ic-17 | ||
Type | Small organic molecule | ||
Emp. Form. | C21H20ClFN4O2 | ||
Mol. Mass. | 414.861 | ||
SMILES | Fc1ccccc1-n1ccc(NC(=O)[C@@H]2CC[C@@H](CC2)Oc2cc(Cl)ccn2)n1 |r,wU:17.21,14.14,(6.42,1.41,;7.19,.08,;8.73,.08,;9.5,-1.26,;8.73,-2.59,;7.19,-2.59,;6.42,-1.26,;4.88,-1.26,;3.97,-2.5,;2.51,-2.03,;2.51,-.49,;1.17,.28,;-.16,-.49,;-.16,-2.03,;-1.49,.28,;-1.49,1.82,;-2.83,2.59,;-4.16,1.82,;-4.16,.28,;-2.83,-.49,;-5.5,2.59,;-6.83,1.82,;-6.83,.28,;-8.16,-.49,;-8.16,-2.03,;-9.5,.28,;-9.5,1.82,;-8.16,2.59,;3.97,-.01,)| | ||
Structure |