| Reaction Details |
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 | Report a problem with these data |
| Target | Cathepsin B |
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| Ligand | BDBM120824 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Enzymatic activity assay |
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| pH | 6±n/a |
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| Temperature | 310.15±n/a K |
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| Ki | 0.668±0.066 nM |
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| Comments | extracted |
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| Citation |  Raghav, N; Garg, S N-formylpyrazolines and N-benzoylpyrazolines as novel inhibitors of mammalian cathepsin B and cathepsin H. Bioorg Chem57:43-50 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cathepsin B |
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| Name: | Cathepsin B |
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| Synonyms: | n/a |
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| Type: | Protein |
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| Mol. Mass.: | 36777.57 |
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| Organism: | Capra hircus (Goat) |
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| Description: | n/a |
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| Residue: | 335 |
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| Sequence: | MWQLLATLSCLLVLTSARSSLHFPPLSDEMVNYVNKQNTTWKAGHNFYNVDLSYVKKLCG
AILGGPKLPQRDAFAADMVLPDSFDAREQWPNCPTIKEIRDQGSCGSCWAFGAVEAISDR
ICIHSKGRVNVEVSAEDMLTCCGSECGDGCNGGFPSGAWNFWTKKGLVSGGLYDSHVGCR
PYSIPPCEHHVNGSRPPCTGEGDTPKCSKICEPGYSPSYKDDKHFGCSSYSVSSNEKEIM
AEIYKNGPVEGAFSVYSDFLLYKSGVYQHVSGEMMGGHAIRILGWGVENDTPYWLVGNSW
NTDWGDKGFFKILRGQDHCGIESEIVAGMPCTHQY
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| BDBM120824 |
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| n/a |
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| Name | BDBM120824 |
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| Synonyms: | N-formyl-5-(-2'-methoxyphenyl)-3-phenylpyrazoline (1e) |
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| Type | Small organic molecule |
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| Emp. Form. | C17H16N2O2 |
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| Mol. Mass. | 280.3211 |
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| SMILES | COc1ccccc1C1CC(=NN1C=O)c1ccccc1 |c:11| |
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| Structure | 
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