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TargetBromodomain-containing protein 4 [368-440]
LigandBDBM50427454
Substrate/Competitorn/a
Meas. Tech.Inhibition Assay
IC50 3451±n/a nM
Citation Durden, DL; Morales, GA; Garlich, JR Thienopyranones as kinase and epigenetic inhibitors US Patent US9505780 Publication Date 11/29/2016
More Info.:Get all data from this article,  Assay Method
 
Bromodomain-containing protein 4 [368-440]
Name:Bromodomain-containing protein 4 [368-440]
Synonyms:BRD4 | BRD4_HUMAN | Bromo domain 2 | Bromodomain-containing protein 4 (BD2) | Bromodomain-containing protein 4 (BRD4) Bromo 2 | Bromodomain-containing protein 4 (BRD4)(BD2) | Bromodomain-containing protein 4 (BRD4)(Bromo 2) | Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2) | Bromodomain-containing protein 4 Bromodomain 2 (BRD4-2) | Bromodomain-containing protein 4 Domain 2 | HUNK1
Type:Protein
Mol. Mass.:8564.63
Organism:Homo sapiens (Human)
Description:BD2 (368-440 aa) of O60885
Residue:73
Sequence:
KHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFS
NCYKYNPPDHEVV
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BDBM50427454
n/a
NameBDBM50427454
Synonyms:CHEMBL2322239 | US10308662, Compound 6 | US9505780, 6
TypeSmall organic molecule
Emp. Form.C17H15NO3S
Mol. Mass.313.371
SMILESO=c1cc(oc2c(csc12)-c1ccccc1)N1CCOCC1
Structure
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