Reaction Details |
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Target | Oxysterols receptor LXR-beta |
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Ligand | BDBM27289 |
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Substrate/Competitor | biotinylated SRC-1 peptide |
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Meas. Tech. | HTRF Cofactor Peptide Recruitment Assay |
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pH | 7.5±n/a |
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Temperature | 295.15±n/a K |
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EC50 | >30000±n/a nM |
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Citation | Bakir, F; Kher, S; Pannala, M; Wilson, N; Nguyen, T; Sircar, I; Takedomi, K; Fukushima, C; Zapf, J; Xu, K; Zhang, SH; Liu, J; Morera, L; Schneider, L; Sakurai, N; Jack, R; Cheng, JF Discovery and structure-activity relationship studies of indole derivatives as liver X receptor (LXR) agonists. Bioorg Med Chem Lett17:3473-9 (2007) [PubMed] Article |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Oxysterols receptor LXR-beta |
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Name: | Oxysterols receptor LXR-beta |
Synonyms: | LXRB | Liver X receptor beta (NR1H2) | Liver X, LXR beta | NER | NR1H2 | NR1H2_HUMAN | Nuclear receptor NER | UNR | Ubiquitously-expressed nuclear receptor |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 50978.79 |
Organism: | Homo sapiens (Human) |
Description: | P55055 |
Residue: | 460 |
Sequence: | MSSPTTSSLDTPLPGNGPPQPGAPSSSPTVKEEGPEPWPGGPDPDVPGTDEASSACSTDW
VIPDPEEEPERKRKKGPAPKMLGHELCRVCGDKASGFHYNVLSCEGCKGFFRRSVVRGGA
RRYACRGGGTCQMDAFMRRKCQQCRLRKCKEAGMREQCVLSEEQIRKKKIRKQQQESQSQ
SQSPVGPQGSSSSASGPGASPGGSEAGSQGSGEGEGVQLTAAQELMIQQLVAAQLQCNKR
SFSDQPKVTPWPLGADPQSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQI
ALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMR
RLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRM
LMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDVHE
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BDBM27289 |
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biotinylated SRC-1 peptide |
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Name: | biotinylated SRC-1 peptide |
Synonyms: | n/a |
Type: | Peptide |
Mol. Mass.: | 3157.52 |
Organism: | n/a |
Description: | A biotinylated peptide comprises amino acids 675-699 of steroid receptor coactivator 1 (SRC1). |
Residue: | 28 |
Sequence: | CPSSHSSLTERHKILHRLLQEGSPS-CONH2
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