| Reaction Details |
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 | Report a problem with these data |
| Target | Chymotrypsin-like elastase family member 2A |
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| Ligand | BDBM50085362 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_152309 |
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| IC50 | 26000±n/a nM |
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| Citation |  Hayashi, Y; Iijima, K; Katada, J; Kiso, Y Structure-activity relationship studies of chloromethyl ketone derivatives for selective human chymase inhibitors. Bioorg Med Chem Lett10:199-201 (2000) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Chymotrypsin-like elastase family member 2A |
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| Name: | Chymotrypsin-like elastase family member 2A |
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| Synonyms: | CEL2A_PIG | CELA2A | ELA2 | ELA2A | Elastase 2A | Elastase-2 | Elastase-2A | Pancreatic elastase |
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| Type: | PROTEIN |
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| Mol. Mass.: | 28705.23 |
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| Organism: | Sus scrofa |
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| Description: | ChEMBL_156951 |
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| Residue: | 269 |
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| Sequence: | MIRALLLSTLVAGALSCGLPANLPQLPRVVGGEDARPNSWPWQVSLQYDSSGQWRHTCGG
TLVDQSWVLTAAHCISSSRTYRVVLGRHSLSTNEPGSLAVKVSKLVVHQDWNSNQLSNGN
DIALLKLASPVSLTDKIQLGCLPAAGTILPNNYVCYVTGWGRLQTNGASPDILQQGQLLV
VDYATCSKPGWWGSTVKTNMICAGGDGIISSCNGDSGGPLNCQGANGQWQVHGIVSFGSS
LGCNYYHKPSVFTRVSNYIDWINSVIANN
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| BDBM50085362 |
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| n/a |
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| Name | BDBM50085362 |
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| Synonyms: | CHEMBL64494 | N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-phenyl-acrylamide |
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| Type | Small organic molecule |
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| Emp. Form. | C19H18ClNO2 |
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| Mol. Mass. | 327.805 |
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| SMILES | ClCC(=O)[C@H](Cc1ccccc1)NC(=O)\C=C\c1ccccc1 |
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| Structure | 
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