| Reaction Details |
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 | Report a problem with these data |
| Target | Ecdysone receptor |
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| Ligand | BDBM50128302 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_65458 |
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| EC50 | 1250±n/a nM |
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| Citation |  Tice, CM; Hormann, RE; Thompson, CS; Friz, JL; Cavanaugh, CK; Saggers, JA Optimization of alpha-acylaminoketone ecdysone agonists for control of gene expression. Bioorg Med Chem Lett13:1883-6 (2003) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Ecdysone receptor |
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| Name: | Ecdysone receptor |
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| Synonyms: | n/a |
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| Type: | PROTEIN |
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| Mol. Mass.: | 57629.46 |
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| Organism: | Choristoneura fumiferana |
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| Description: | ChEMBL_65458 |
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| Residue: | 513 |
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| Sequence: | MDLKHEVAYRGVLPGQVKAEPGVHNGQVNGHVRDWMAGGAGANSPSPGAVAQPQPNNGYS
SPLSSGSYGPYSPNGKIGREELSPASSINGCSTDGEARRQKKGPAPRQQEELCLVCGDRA
SGYHYNALTCEGCKGFFRRSVTKNAVYICKFGHACEMDMYMRRKCQECRLKKCLAVGMRP
ECVVPETQCAMKRKEKKAQKEKDKLPVSTTTVDDHMPPIMQCEPPPPEAARIHEVVPRFL
SDKLLETNRQKNIPQLTANQQFLIARLIWYQDGYEQPSDEDLKRITQTWQQADDENEESD
TPFRQITEMTILTVQLIVEFAKGLPGFAKISQPDQITLLKACSSEVMMLRVARRYDAASD
SVLFANNQAYTRDNYRKAGMAYVIEDLLHFCRCMYSMALDNIHYALLTAVVIFSDRPGLE
QPQLVEEIQRYYLNTLRIYILNQLSGSARSSVIYGKILSILSELRTLGMQNSNMCISLKL
KNRKLPPFLEEIWDVADMSHTQPPPILESPTNL
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| BDBM50128302 |
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| n/a |
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| Name | BDBM50128302 |
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| Synonyms: | CHEMBL59044 | N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-2-ethyl-3-methoxy-benzamide |
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| Type | Small organic molecule |
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| Emp. Form. | C25H31NO3 |
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| Mol. Mass. | 393.5185 |
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| SMILES | CCc1c(OC)cccc1C(=O)NC1(CCCCC1)C(=O)c1cc(C)cc(C)c1 |
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| Structure | 
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