| Reaction Details |
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 | Report a problem with these data |
| Target | Melanocortin receptor 4 |
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| Ligand | BDBM135734 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Competitive Binding Assay Using Eu-NDP-a-MSH |
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| Temperature | 310.15±n/a K |
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| Ki | 3±n/a nM |
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| Comments | extracted |
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| Citation |  Shi, Y; Sharma, SD; Dodd, JH; Yang, W Melanocortin receptor-specific heptapeptides US Patent US9458201 Publication Date 10/4/2016 |
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| More Info.: | Get all data from this article, Assay Method |
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| Melanocortin receptor 4 |
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| Name: | Melanocortin receptor 4 |
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| Synonyms: | MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R) |
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| Type: | Enzyme |
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| Mol. Mass.: | 36949.50 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P32245 |
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| Residue: | 332 |
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| Sequence: | MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLL
ENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVN
IDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVS
GILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGAN
MKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPL
IYALRSQELRKTFKEIICCYPLGGLCDLSSRY
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| BDBM135734 |
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| n/a |
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| Name | BDBM135734 |
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| Synonyms: | US10179804, Example 119 | US10632171, Peptide No. 119 | US8846601, 119 | US9458201, 119 |
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| Type | Small organic molecule |
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| Emp. Form. | C48H71N17O9 |
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| Mol. Mass. | 1030.1858 |
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| SMILES | CC(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@H]1CCCNC(=O)CC[C@H](NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](CCN)NC1=O)C(N)=O |r| |
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| Structure | 
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