| Reaction Details |
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 | Report a problem with these data |
| Target | Low molecular weight phosphotyrosine protein phosphatase |
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| Ligand | BDBM533325 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | LMPTP Primary Screening Protocol |
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| IC50 | 500±n/a nM |
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| Citation |  Bottini, N; Zou, J; Ganji, SR; Stanford, S; Pinkerton, A; Chung, TD; Hedrick, M; Ardecky, R Inhibitors of low molecular weight protein tyrosine phosphatase and uses thereof US Patent US11220486 Publication Date 1/11/2022 |
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| More Info.: | Get all data from this article, Assay Method |
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| Low molecular weight phosphotyrosine protein phosphatase |
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| Name: | Low molecular weight phosphotyrosine protein phosphatase |
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| Synonyms: | 3.1.3.2 | 3.1.3.48 | ACP1 | Adipocyte acid phosphatase | LMW-PTP | LMW-PTPase | LMWPTP | Low molecular weight cytosolic acid phosphatase | PPAC_HUMAN | Red cell acid phosphatase 1 | low molecular weight phosphotyrosine protein phosphatase isoform c |
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| Type: | n/a |
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| Mol. Mass.: | 18042.81 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P24666 |
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| Residue: | 158 |
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| Sequence: | MAEQATKSVLFVCLGNICRSPIAEAVFRKLVTDQNISENWRVDSAATSGYEIGNPPDYRG
QSCMKRHGIPMSHVARQITKEDFATFDYILCMDESNLRDLNRKSNQVKTCKAKIELLGSY
DPQKQLIIEDPYYGNDSDFETVYQQCVRCCRAFLEKAH
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| BDBM533325 |
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| n/a |
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| Name | BDBM533325 |
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| Synonyms: | N-[(4-{4-[(3-piperidylpropyl)amino]-2- quinolyl}phenyl)methyl]acetamide | US10626094, Example I255 | US11220486, Compound I255 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H32N4O |
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| Mol. Mass. | 416.5585 |
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| SMILES | CC(=O)NCc1ccc(cc1)-c1cc(NCCCC2CCCNC2)c2ccccc2n1 |
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| Structure | 
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