| Reaction Details |
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 | Report a problem with these data |
| Target | Glucagon-like peptide 1 receptor |
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| Ligand | BDBM620514 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | The Alizarin Assay (ARS) (Glucose) |
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| Kd | 1700000±n/a nM |
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| Citation |  Kruse, T; Kofod-Hansen, M; Muenzel, MW; Thoegersen, H; Sauerberg, P; Rasmussen, JE; Behrens, C; Hoeg-Jensen, T; Balsanek, V; Drobnakova, Z; Droz, L; Havranek, M; Kotek, V; Stengl, M; Snajdr, I; Drusanova, H Glucose-sensitive albumin-binding derivatives US Patent US11767332 Publication Date 9/26/2023 |
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| More Info.: | Get all data from this article, Assay Method |
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| Glucagon-like peptide 1 receptor |
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| Name: | Glucagon-like peptide 1 receptor |
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| Synonyms: | GLP-1 receptor | GLP-1-R | GLP-1R | GLP1R | GLP1R_HUMAN | Glucagon-like peptide 1 receptor | Glucagon-like peptide 1 receptor (GLP-1) |
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| Type: | Enzyme |
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| Mol. Mass.: | 53035.78 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P43220 |
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| Residue: | 463 |
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| Sequence: | MAGAPGPLRLALLLLGMVGRAGPRPQGATVSLWETVQKWREYRRQCQRSLTEDPPPATDL
FCNRTFDEYACWPDGEPGSFVNVSCPWYLPWASSVPQGHVYRFCTAEGLWLQKDNSSLPW
RDLSECEESKRGERSSPEEQLLFLYIIYTVGYALSFSALVIASAILLGFRHLHCTRNYIH
LNLFASFILRALSVFIKDAALKWMYSTAAQQHQWDGLLSYQDSLSCRLVFLLMQYCVAAN
YYWLLVEGVYLYTLLAFSVLSEQWIFRLYVSIGWGVPLLFVVPWGIVKYLYEDEGCWTRN
SNMNYWLIIRLPILFAIGVNFLIFVRVICIVVSKLKANLMCKTDIKCRLAKSTLTLIPLL
GTHEVIFAFVMDEHARGTLRFIKLFTELSFTSFQGLMVAILYCFVNNEVQLEFRKSWERW
RLEHLHIQRDSSMKPLKCPTSSLSSGATAGSSMYTATCQASCS
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| BDBM620514 |
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| n/a |
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| Name | BDBM620514 |
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| Synonyms: | (3-Borono-5-((3-borono-5-(trifluoromethyl)phenyl)sulfonyl)glycine | US11767332, Example 20 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H14B2F3NO9S |
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| Mol. Mass. | 474.966 |
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| SMILES | OB(O)c1cc(cc(c1)S(=O)(=O)c1cc(cc(c1)C(F)(F)F)B(O)O)C(=O)NCC(O)=O |
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| Structure | 
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