Reaction Details |
| Report a problem with these data |
Target | Somatostatin receptor type 1 |
---|
Ligand | BDBM311920 |
---|
Substrate/Competitor | n/a |
---|
Meas. Tech. | Radioligand Binding Assay |
---|
Ki | 3460±n/a nM |
---|
Citation | Giovannini, R; Cui, Y; Doods, H; Ferrara, M; Just, S; Kuelzer, R; Lingard, I; Mazzaferro, R; Rudolf, K Somatostatin receptor subtype 4 (SSTR4) agonists US Patent US9789082 Publication Date 10/17/2017 |
---|
More Info.: | Get all data from this article, Assay Method |
---|
|
Somatostatin receptor type 1 |
---|
Name: | Somatostatin receptor type 1 |
Synonyms: | SOMATOSTATIN SST1 | SRIF-2 | SS-1-R | SS1-R | SS1R | SSR1_HUMAN | SSTR1 | Somatostatin receptor type 1 (SSTR1) |
Type: | Enzyme |
Mol. Mass.: | 42692.81 |
Organism: | Homo sapiens (Human) |
Description: | P30872 |
Residue: | 391 |
Sequence: | MFPNGTASSPSSSPSPSPGSCGEGGGSRGPGAGAADGMEEPGRNASQNGTLSEGQGSAIL
ISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLL
RHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLG
VWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAIC
LCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQD
DATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKS
RAYSVEDFQPENLESGGVFRNGTCTSRITTL
|
|
|
BDBM311920 |
---|
n/a |
---|
Name | BDBM311920 |
Synonyms: | US10166214, Example 56 | US10675268, Example 56 | US9789082, Example 56 |
Type | Small organic molecule |
Emp. Form. | C19H23N3O2 |
Mol. Mass. | 325.4048 |
SMILES | CC(C)(COc1nccc2ccccc12)NC(=O)[C@@H]1[C@H]2CNC[C@@H]12 |r| |
Structure |
|