Reaction Details |
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Target | Somatostatin receptor type 1 |
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Ligand | BDBM311971 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Radioligand Binding Assay |
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Ki | 4300±n/a nM |
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Citation | Giovannini, R; Cui, Y; Doods, H; Ferrara, M; Just, S; Kuelzer, R; Lingard, I; Mazzaferro, R; Rudolf, K Somatostatin receptor subtype 4 (SSTR4) agonists US Patent US9789082 Publication Date 10/17/2017 |
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More Info.: | Get all data from this article, Assay Method |
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Somatostatin receptor type 1 |
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Name: | Somatostatin receptor type 1 |
Synonyms: | SOMATOSTATIN SST1 | SRIF-2 | SS-1-R | SS1-R | SS1R | SSR1_HUMAN | SSTR1 | Somatostatin receptor type 1 (SSTR1) |
Type: | Enzyme |
Mol. Mass.: | 42692.81 |
Organism: | Homo sapiens (Human) |
Description: | P30872 |
Residue: | 391 |
Sequence: | MFPNGTASSPSSSPSPSPGSCGEGGGSRGPGAGAADGMEEPGRNASQNGTLSEGQGSAIL
ISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLL
RHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLG
VWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAIC
LCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQD
DATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKS
RAYSVEDFQPENLESGGVFRNGTCTSRITTL
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BDBM311971 |
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n/a |
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Name | BDBM311971 |
Synonyms: | US10166214, Example 107 | US10675268, Example 107 | US9789082, Example 107 |
Type | Small organic molecule |
Emp. Form. | C18H24N4O |
Mol. Mass. | 312.4094 |
SMILES | Cc1cccc2c(nn(C)c12)C(C)(C)NC(=O)[C@@H]1[C@H]2CNC[C@@H]12 |r| |
Structure |
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