| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 3 |
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| Ligand | BDBM50081059 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Radioligand Binding Assay |
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| Ki | >8710±n/a nM |
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| Citation |  Giovannini, R; Cui, Y; Doods, H; Ferrara, M; Just, S; Kuelzer, R; Lingard, I; Mazzaferro, R; Rudolf, K Somatostatin receptor subtype 4 (SSTR4) agonists US Patent US9789082 Publication Date 10/17/2017 |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 3 |
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| Name: | Somatostatin receptor type 3 |
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| Synonyms: | SOMATOSTATIN SST3 | SS-3-R | SS3-R | SS3R | SSR-28 | SSR3_HUMAN | SSTR3 | Somatostatin receptor type 3 (SSTR3) |
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| Type: | Protein |
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| Mol. Mass.: | 45855.97 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P32745 |
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| Residue: | 418 |
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| Sequence: | MDMLHPSSVSTTSEPENASSAWPPDATLGNVSAGPSPAGLAVSGVLIPLVYLVVCVVGLL
GNSLVIYVVLRHTASPSVTNVYILNLALADELFMLGLPFLAAQNALSYWPFGSLMCRLVM
AVDGINQFTSIFCLTVMSVDRYLAVVHPTRSARWRTAPVARTVSAAVWVASAVVVLPVVV
FSGVPRGMSTCHMQWPEPAAAWRAGFIIYTAALGFFGPLLVICLCYLLIVVKVRSAGRRV
WAPSCQRRRRSERRVTRMVVAVVALFVLCWMPFYVLNIVNVVCPLPEEPAFFGLYFLVVA
LPYANSCANPILYGFLSYRFKQGFRRVLLRPSRRVRSQEPTVGPPEKTEEEDEEEEDGEE
SREGGKGKEMNGRVSQITQPGTSGQERPPSRVASKEQQLLPQEASTGEKSSTMRISYL
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| BDBM50081059 |
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| n/a |
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| Name | BDBM50081059 |
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| Synonyms: | CHEMBL3421845 | US10166214, Example 138 | US10675268, Example 138 | US9789082, Example 138 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H22N4O |
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| Mol. Mass. | 310.3935 |
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| SMILES | [H][C@@]12CNC[C@]1([H])[C@H]2C(=O)NC(C)(C)c1nc(C)nc2ccccc12 |r| |
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| Structure | 
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