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TargetVascular endothelial growth factor A
LigandBDBM373005
Substrate/Competitorn/a
Meas. Tech.ELISA Assay
EC50 7.00±n/a nM
Citation Dixon, DDGrina, JJosey, JARizzi, JPSchlachter, STWallace, EMWang, BWehn, PXu, RYang, H Aryl ethers and uses thereof US Patent US9896418 Publication Date 2/20/2018
More Info.:Get all data from this article,  Assay Method
 
Vascular endothelial growth factor A
Name:Vascular endothelial growth factor A
Synonyms:VEGF | VEGF-A | VEGFA | VEGFA_HUMAN | VPF | Vascular endothelial growth factor (VEGF) | Vascular endothelial growth factor A (VEGF) | Vascular endothelial growth factor A (VEGF2) | Vascular permeability factor
Type:Protein
Mol. Mass.:27063.81
Organism:Homo sapiens (Human)
Description:P15692
Residue:395
Sequence:
MTDRQTDTAPSPSYHLLPGRRRTVDAAASRGQGPEPAPGGGVEGVGARGVALKLFVQLLG
CSRFGGAVVRAGEAEPSGAARSASSGREEPQPEEGEEEEEKEEERGPQWRLGARKPGSWT
GEAAVCADSAPAARAPQALARASGRGGRVARRGAEESGPPHSPSRRGSASRAGPGRASET
MNFLLSWVHWSLALLLYLHHAKWSQAAPMAEGGGQNHHEVVKFMDVYQRSYCHPIETLVD
IFQEYPDEIEYIFKPSCVPLMRCGGCCNDEGLECVPTEESNITMQIMRIKPHQGQHIGEM
SFLQHNKCECRPKKDRARQEKKSVRGKGKGQKRKRKKSRYKSWSVPCGPCSERRKHLFVQ
DPQTCKCSCKNTDSRCKARQLELNERTCRCDKPRR
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BDBM373005
n/a
NameBDBM373005
Synonyms:US10597366, Compound 159 | US9896418, Compound 159
TypeSmall organic molecule
Emp. Form.C16H12F4O4S
Mol. Mass.376.323
SMILESCS(=O)(=O)c1ccc(Oc2cc(F)cc(F)c2)c2CC(F)(F)C(O)c12
Structure
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